SCHEMBL29907757

SCHEMBL29907757

Cc1ccc(-c2ncc(C(N)=O)nc2-c2ccc(=O)n(C)c2)o1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 13/20 0.48
ADORA1 P30542 6/20 0.48
ADORA3 P0DMS8 3/20 0.48
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
PKM P14618 1/20 0.39
ADORA2B P29275 3/20 0.39
DGAT1 O75907 1/20 0.35
SOAT1 P35610 1/20 0.35
CNR1 P21554 1/20 0.34
BRD4 O60885 1/20 0.34
ATR Q13535 1/20 0.34
DYRK1A Q13627 1/20 0.34
MEN1 O00255 1/20 0.34
USP2 O75604 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
RECQL P46063 1/20 0.34
KMT2A Q03164 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28463384 0.81 ADORA2A (0.55) ADORA2AADORA1ADORA3ADORA2BBRD4
SCHEMBL29907659 0.80 ADORA2A (0.56) ADORA2AADORA1ADORA3ADORA2BCNR1
SCHEMBL29907672 0.78 ADORA2A (0.51) ADORA2AADORA1ADORA2BBRD4DYRK1A
SCHEMBL22552045 0.77 ADORA2A (0.47) ADORA2AADORA1ADORA3KDM4EALDH1A1
SCHEMBL29907698 0.77 ADORA2A (0.47) ADORA2AADORA1ADORA3KDM4EALDH1A1
SCHEMBL22579112 0.75 ADORA2A (0.49) ADORA2AADORA1ADORA3KDM4EALDH1A1
SCHEMBL29907681 0.75 ADORA2A (0.48) ADORA2AADORA1ADORA2BDGAT1SOAT1
SCHEMBL22579156 0.73 ADORA2A (0.48) ADORA2AADORA1ADORA3ADORA2BBRD4
SCHEMBL13680725 0.72 ADORA2A (0.51) ADORA2AADORA1ADORA3KDM4EALDH1A1
SCHEMBL22579095 0.68 ADORA2A (0.51) ADORA2AADORA1ADORA3ADORA2BATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115181092-A Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2022-10-14 CN disclosed
CN-112279837-B Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2022-08-09 CN disclosed