SCHEMBL13680736

SCHEMBL13680736

CC(=O)Cn1cc(-c2nc(C)cs2)cn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.39
CYP2E1 P05181 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2A6 P11509 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2B6 P20813 1/20 0.39
ALDH1A1 P00352 1/20 0.37
EIF2AK2 P19525 1/20 0.37
TGFBR1 P36897 2/20 0.37
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
TSHR P16473 1/20 0.36
AOC3 Q16853 2/20 0.35
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
S1PR1 P21453 1/20 0.34
KDM4E B2RXH2 1/20 0.34
USP2 O75604 1/20 0.34
ALOX15 P16050 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13681048 0.79 BTK (0.36) BTKALDH1A1EIF2AK2RAB9ASMN1; SMN2
SCHEMBL19002406 0.72 CYP3A4 (0.47) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL13680671 0.72 CYP2A6 (0.44) BTKCYP2A6ALDH1A1TGFBR1KDM4E
SCHEMBL6938232 0.70 ALPI (0.54) CYP3A4CYP2C9ALDH1A1RAB9ASMN1; SMN2
SCHEMBL13680749 0.69 ALDH1A1 (0.46) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL13680646 0.68 EIF2AK2 (0.46) EIF2AK2GRIN1GRIN2B
SCHEMBL13680717 0.68 FGFR1 (0.40) BTKCYP2C9ALDH1A1RAB9ASMN1; SMN2
SCHEMBL13680742 0.67 CYP2E1 (0.45) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL16437820 0.65 ALDH1A1 (0.45) ALDH1A1TSHRRAB9ASMN1; SMN2S1PR1
SCHEMBL13113429 0.65 HSD17B10 (0.50) ALDH1A1RAB9ASMN1; SMN2S1PR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed