SCHEMBL13680749

SCHEMBL13680749

CC(=O)Cc1ccc(-c2nc(C)cs2)cc1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
RAB9A P51151 4/20 0.46
NPC1 O15118 2/20 0.46
PPARA Q07869 2/20 0.46
AOC3 Q16853 2/20 0.44
CYP2E1 P05181 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2A6 P11509 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2B6 P20813 1/20 0.44
KDM4E B2RXH2 1/20 0.43
HPGD P15428 1/20 0.43
POLB P06746 2/20 0.43
LMNA P02545 2/20 0.43
GAA P10253 2/20 0.39
MEN1 O00255 1/20 0.39
THRB P10828 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8198560 0.80 CYP3A4 (0.60) ALDH1A1RAB9ANPC1AOC3CYP2E1
SCHEMBL13680487 0.80 ALDH1A1 (0.49) ALDH1A1RAB9ANPC1PPARAAOC3
SCHEMBL8021391 0.80 CYP3A4 (0.49) ALDH1A1RAB9ANPC1PPARAAOC3
SCHEMBL7905176 0.78 CYP3A4 (0.58) ALDH1A1RAB9ANPC1AOC3CYP2E1
SCHEMBL23328877 0.78 RAB9A (0.60) ALDH1A1RAB9ANPC1PPARAAOC3
SCHEMBL13680478 0.77 KDM4E (0.62) ALDH1A1RAB9ANPC1PPARAKDM4E
Acetic Acid SCHEMBL5472574 0.77 CYP2E1 (0.54) ALDH1A1RAB9ANPC1CYP2E1CYP3A4
SCHEMBL13680525 0.76 RAB9A (0.49) ALDH1A1RAB9ANPC1PPARAAOC3
SCHEMBL13680522 0.76 RAB9A (0.55) ALDH1A1RAB9ANPC1KDM4EHPGD
SCHEMBL21873479 0.76 RAB9A (0.54) ALDH1A1RAB9ANPC1PPARAAOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed