SCHEMBL13680750

SCHEMBL13680750

Cc1csc(-c2cnc(=O)n(C)c2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.44
ADORA1 P30542 1/20 0.44
CYP3A4 P08684 2/20 0.43
CYP2E1 P05181 1/20 0.43
CYP2A6 P11509 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2B6 P20813 1/20 0.43
GABRA1 P14867 6/20 0.40
GABRG2 P18507 6/20 0.40
GABRB3 P28472 6/20 0.40
GABRA3 P34903 6/20 0.40
GABRA2 P47869 5/20 0.40
GABRA5 P31644 4/20 0.40
GRIN1 Q05586 1/20 0.39
GRIN2B Q13224 1/20 0.39
PDE10A Q9Y233 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680757 0.76 ADORA2A (0.56) ADORA2AADORA1CYP3A4CYP2E1CYP2A6
SCHEMBL13681064 0.76 LMNA (0.39) PDE10AKDM4EALDH1A1TP53HPGD
SCHEMBL19002406 0.73 CYP3A4 (0.47) ADORA2AADORA1CYP3A4CYP2E1CYP2A6
SCHEMBL13680744 0.72 CYP3A4 (0.53) ADORA2AADORA1CYP3A4CYP2E1CYP2A6
SCHEMBL13680755 0.70 CYP2E1 (0.44) ADORA2AADORA1CYP3A4CYP2E1CYP2A6
SCHEMBL6840352 0.69 CYP3A4 (0.64) CYP3A4CYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL13680738 0.69 CYP3A4 (0.50) ADORA2AADORA1CYP3A4CYP2E1CYP2A6
SCHEMBL13680689 0.69 CYP2A6 (0.49) ADORA2AADORA1CYP2A6TGFBR1
SCHEMBL13680739 0.68 ADORA2A (0.49) ADORA2AADORA1CYP3A4CYP2E1CYP2A6
SCHEMBL13680742 0.68 CYP2E1 (0.45) CYP3A4CYP2E1CYP2A6CYP2C9CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed