SCHEMBL13680755

SCHEMBL13680755

Cc1csc(-c2cnc(=O)[nH]c2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2E1 P05181 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2A6 P11509 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2B6 P20813 1/20 0.44
EIF4E P06730 1/20 0.42
PDE10A Q9Y233 1/20 0.38
GLA P06280 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
TGFBR1 P36897 3/20 0.35
BMPR1A P36894 1/20 0.35
SMAD2 Q15796 1/20 0.35
PIK3CA P42336 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3550642 0.75 KMT2A (0.49) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL13680744 0.73 CYP3A4 (0.53) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL6885089 0.71 SMN1; SMN2 (0.40) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL6840352 0.70 CYP3A4 (0.64) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL13680738 0.70 CYP3A4 (0.50) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL13680750 0.70 ADORA2A (0.44) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL13680739 0.69 ADORA2A (0.49) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL13680742 0.69 CYP2E1 (0.45) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL8198560 0.68 CYP3A4 (0.60) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL13680746 0.68 CYP3A4 (0.47) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed