SCHEMBL13683254

SCHEMBL13683254

COc1ccc(NS(=O)(=O)c2sc3ccc(C)cc3c2C)cc1N1CCNCC1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 19/20 0.83
HTR1A P08908 8/20 0.83
HTR1D P28221 8/20 0.83
HTR1B P28222 8/20 0.83
HTR2C P28335 6/20 0.83
DRD2 P14416 6/20 0.83
ADRA1B P35368 6/20 0.83
DRD3 P35462 6/20 0.83
HTR7 P34969 5/20 0.83
HTR4 Q13639 5/20 0.83
HTR2A P28223 5/20 0.83
DRD1 P21728 1/20 0.83
DRD4 P21917 1/20 0.83
HTR2B P41595 5/20 0.82
CYP1A2 P05177 1/20 0.82
ADRB1 P08588 1/20 0.82
CYP3A4 P08684 1/20 0.82
ADRA2A P08913 1/20 0.82
CYP2D6 P10635 1/20 0.82
ADRB3 P13945 1/20 0.82

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29386932 0.91 HTR6 (1.00) HTR6HTR1AHTR1DHTR1BHTR2C
SCHEMBL194700 0.91 HTR6 (1.00) HTR6HTR1AHTR1DHTR1BHTR2C
Hydrochloric Acid SCHEMBL6977773 0.90 HTR6 (1.00) HTR6HTR1AHTR1DHTR1BHTR2C
SCHEMBL29496144 0.81 HTR6 (1.00) HTR6HTR1AHTR1DHTR1BHTR2C
SCHEMBL1136525 0.81 HTR6 (1.00) HTR6HTR1AHTR1DHTR1BHTR2C
SCHEMBL7199110 0.79 HTR6 (0.82) HTR6HTR1AHTR1DHTR1BHTR2C
SCHEMBL194699 0.77 HTR6 (0.76) HTR6HTR1AHTR1DHTR1BHTR2C
SCHEMBL4801548 0.77 GHSR (1.00) HTR6HTR1AHTR1DHTR1BHTR2C
SCHEMBL4801555 0.77 GHSR (1.00) HTR6HTR1AHTR1DHTR1BHTR2C
SCHEMBL6983122 0.76 HTR6 (0.65) HTR6HTR1AHTR1DHTR1BHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7592457-B2 3-aryl-3-methyl-quinoline-2, 4-diones, preparation method thereof, and pharmaceutical composition containing the same KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2009-09-22 US disclosed