SCHEMBL13683402

SCHEMBL13683402

CN(Cc1ccncc1)CC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
LOXL2 Q9Y4K0 2/20 0.37
CHRM5 P08912 1/20 0.37
CHKA P35790 1/20 0.37
CYP1A2 P05177 3/20 0.37
CYP3A4 P08684 3/20 0.37
CYP2D6 P10635 3/20 0.37
CYP2C9 P11712 3/20 0.37
CYP2C19 P33261 3/20 0.37
ALOX15 P16050 1/20 0.37
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
ALDH1A1 P00352 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PYCR1 P32322 1/20 0.35
MMP13 P45452 1/20 0.35
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27947483 0.83 SMN1; SMN2 (0.50) KDM4ESMN1; SMN2CHRNB2CHRNA4LOXL2
SCHEMBL30093206 0.81 KDM4E (0.53) KDM4ESMN1; SMN2CHRNB2CHRNA4LOXL2
SCHEMBL9281673 0.79 ALDH1A1 (0.54) KDM4ESMN1; SMN2CYP3A4ALDH1A1PYCR1
SCHEMBL13683403 0.78 CHRNB2 (0.69) KDM4ECHRNB2CHRNA4CYP1A2CYP2D6
SCHEMBL25541294 0.78 KDM4E (0.42) KDM4ECYP2D6ALDH1A1PYCR1
SCHEMBL13239689 0.77 ALDH1A1 (0.44) KDM4ESMN1; SMN2CHRM5CYP1A2CYP3A4
SCHEMBL733206 0.77 CHRNB2 (0.62) KDM4ESMN1; SMN2CHRNB2CHRNA4CHRM5
SCHEMBL25530530 0.76 LMNA (0.51) CYP1A2CYP2D6CYP2C19PYCR1RAB9A
SCHEMBL24368300 0.75 KDM4E (0.45) KDM4ESMN1; SMN2CHRNB2CHRNA4LOXL2
SCHEMBL14432093 0.75 CHRM5 (0.44) KDM4ESMN1; SMN2CHRNB2CHRNA4LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7592373-B2 Amide compounds with MCH antagonistic activity and medicaments comprising these compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-09-22 US disclosed
US-7592373-B2 Amide compounds with MCH antagonistic activity and medicaments comprising these compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-09-22 US disclosed