SCHEMBL13686394

SCHEMBL13686394

COc1ccc(Cl)c(N=O)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.41
ALDH1A1 P00352 4/20 0.40
KDM4E B2RXH2 2/20 0.40
KMT2A Q03164 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
APOBEC3G Q9HC16 2/20 0.39
APOBEC3A P31941 1/20 0.39
ERN1 O75460 1/20 0.39
TRIM24 O15164 1/20 0.39
TYR P14679 1/20 0.39
TRIM33 Q9UPN9 1/20 0.39
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA7 P43166 2/20 0.39
CA9 Q16790 2/20 0.39
CA14 Q9ULX7 2/20 0.39
MAPT P10636 3/20 0.39
MPI P34949 2/20 0.39
TYK2 P29597 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3951891 0.82 CA12 (0.40) TDP1ALDH1A1KDM4EKMT2AAPOBEC3G
SCHEMBL11933957 0.81 CYP1B1 (0.44) ALDH1A1KDM4EKMT2AAPOBEC3GAPOBEC3A
SCHEMBL7774163 0.79 ALDH1A1 (0.46) TDP1ALDH1A1KDM4EKMT2AAPOBEC3G
SCHEMBL30892213 0.78 CA12 (0.56) ALDH1A1KDM4EKMT2AL3MBTL1APOBEC3G
SCHEMBL12878065 0.78 MPI (0.46) ALDH1A1KDM4EL3MBTL1APOBEC3GAPOBEC3A
SCHEMBL12463621 0.78 CA12 (0.56) ALDH1A1KDM4EKMT2AL3MBTL1APOBEC3G
SCHEMBL12878040 0.77 ALDH1A1 (0.59) ALDH1A1KDM4EKMT2AL3MBTL1ERN1
SCHEMBL10967015 0.77 APLNR (0.41) TDP1ALDH1A1KDM4EKMT2AAPOBEC3G
SCHEMBL13266801 0.76 OPRD1 (0.42) ALDH1A1KDM4EKMT2AL3MBTL1APOBEC3G
SCHEMBL13636916 0.76 APOBEC3A (0.39) ALDH1A1KDM4EKMT2AAPOBEC3GAPOBEC3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2103596-A1 Process for the preparation of N-(phenylethyl) anilines salts and solvates thereof useful as serotonin 5-HT6 antagonists Laboratorios Del. Dr. Esteve, S.A. (ES) 2009-09-23 EP disclosed
US-7528163-B2 N,N-Dibutyl-2-[3-(2,2-dimethylpropanoyl)-6-methoxy-1H-indazol-1-yl]acetamide; potassium channel blocker; eye neuroprotectant; hypotensive agent; glaucoma, intraoccular pressure in the eye MERCK & CO. INC. (US) 2009-05-05 US disclosed
US-7410992-B2 Ophthalmic compositions for treating ocular hypertension MERCK & CO. INC. (US) 2008-08-12 US disclosed