SCHEMBL13686454

SCHEMBL13686454

CC1CCc2c(N)ncnc2N1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LIMK1 P53667 5/20 0.40
NNMT P40261 2/20 0.37
KDR P35968 5/20 0.33
CHEK1 O14757 2/20 0.33
DAPK3 O43293 2/20 0.33
PRKD3 O94806 2/20 0.33
MAP4K4 O95819 2/20 0.33
RET P07949 2/20 0.33
FGFR1 P11362 2/20 0.33
FLT1 P17948 2/20 0.33
LTK P29376 2/20 0.33
GRK5 P34947 2/20 0.33
CSNK1A1 P48729 2/20 0.33
CDK8 P49336 2/20 0.33
CDK7 P50613 2/20 0.33
RPS6KA3 P51812 2/20 0.33
CDK5 Q00535 2/20 0.33
TYRO3 Q06418 2/20 0.33
LRRK2 Q5S007 2/20 0.33
AURKB Q96GD4 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13686448 0.71 HTR2C (0.41)
SCHEMBL2606409 0.68 KDR (0.50) LIMK1NNMTKDRCHEK1DAPK3
SCHEMBL30159408 0.68 KDR (0.50) LIMK1NNMTKDRCHEK1DAPK3
SCHEMBL30278084 0.68 DGAT1 (0.35) LIMK1NNMTKDRCHEK1DAPK3
SCHEMBL17362743 0.66 KDR (0.47) LIMK1NNMTKDRCHEK1DAPK3
SCHEMBL20731022 0.64 NNMT (0.43) NNMT
SCHEMBL18297361 0.64 KDR (0.42) LIMK1KDRCHEK1DAPK3PRKD3
SCHEMBL17690273 0.63 LIMK1 (0.50) LIMK1
SCHEMBL24954034 0.62 KDR (0.40) LIMK1KDRCHEK1DAPK3PRKD3
SCHEMBL30159493 0.62 KDR (0.40) LIMK1KDRCHEK1DAPK3PRKD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009107767-A1 NOVEL BICYCLIC PYRIMIDINE DERIVATIVE HAVING ANTAGONISTIC ACTIVITY ON H4 RECEPTOR 大日本住友製薬株式会社 (JP) 2009-09-03 WO disclosed