SCHEMBL1370441

SCHEMBL1370441

CC(C)(C)c1cc2ccccc2c(N)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.46
NCF1 P14598 2/20 0.42
BACE1 P56817 2/20 0.42
F12 P00748 1/20 0.42
PLAU P00749 1/20 0.42
NOS3 P29474 1/20 0.42
NOS1 P29475 1/20 0.42
NOS2 P35228 1/20 0.42
DCPS Q96C86 1/20 0.38
HSD17B10 Q99714 2/20 0.38
KDM4E B2RXH2 2/20 0.37
CYP1B1 Q16678 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP1A1 P04798 1/20 0.37
CCR4 P51679 2/20 0.36
ALDH1A1 P00352 2/20 0.36
GAA P10253 2/20 0.36
HIF1A Q16665 1/20 0.35
HTR2A P28223 1/20 0.35
CYP2A6 P11509 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12145214 0.81 KDM4E (0.46) HTR3ANCF1BACE1F12PLAU
SCHEMBL31631613 0.81 KDM4E (0.46) HTR3ANCF1BACE1F12PLAU
SCHEMBL24995419 0.78 TSHR (0.38) HSD17B10CYP1B1CYP1A2CCR4ALDH1A1
SCHEMBL10220781 0.78 CYP2A6 (0.44) HSD17B10KDM4ECYP1B1CYP1A2CCR4
SCHEMBL15427884 0.77 CCR4 (0.36) HSD17B10CYP1B1CYP1A2CCR4ALDH1A1
SCHEMBL24174415 0.75 SYK (0.50) NOS3NOS1NOS2DCPSHSD17B10
SCHEMBL24174649 0.74 ATM (0.36) HSD17B10CYP1B1CYP1A2CCR4ALDH1A1
SCHEMBL25465465 0.74 HMGCR (0.38) HSD17B10KDM4ECYP1B1CYP1A2CCR4
SCHEMBL5529985 0.74 ADORA2A (0.47) HTR3AKDM4ECCR4ALDH1A1LMNA
SCHEMBL5034624 0.74 NCF1 (0.52) HTR3ANCF1BACE1F12PLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022002118-A1 FUSED-RING HETEROCYCLE DERIVATIVE AND MEDICAL USE THEREOF 四川海思科制药有限公司 2022-01-06 WO disclosed
US-20170309832-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2017-10-26 US disclosed
US-20170309832-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2017-10-26 US disclosed
US-9673402-B2 Platinum metal complexes with divalent groups bridging two ligands MERCK PATENT GMBH (DE) 2017-06-06 US disclosed
US-9673402-B2 Platinum metal complexes with divalent groups bridging two ligands MERCK PATENT GMBH (DE) 2017-06-06 US disclosed
US-9273080-B2 Metal complexes MEREK PATENT GMBH (DE) 2016-03-01 US disclosed
US-9273080-B2 Metal complexes MEREK PATENT GMBH (DE) 2016-03-01 US disclosed
US-9169282-B2 Metal complexes MERCK PATENT GMBH (DE) 2015-10-27 US disclosed
US-9169282-B2 Metal complexes MERCK PATENT GMBH (DE) 2015-10-27 US disclosed
US-9169282-B2 Metal complexes MERCK PATENT GMBH (DE) 2015-10-27 US disclosed
EP-2726490-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2015-04-29 EP disclosed
US-20130082209-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2013-04-04 US disclosed
US-20130082209-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2013-04-04 US disclosed
WO-2013000531-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2013-01-03 WO disclosed
WO-2011157339-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2011-12-22 WO disclosed
US-20110284799-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2011-11-24 US disclosed
US-20110284799-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2011-11-24 US disclosed
US-20110284799-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2011-11-24 US disclosed
WO-2010086089-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2010-08-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110284799-A1 METAL COMPLEXES SOD1, AP1M1, AP3M1 HTR3A 4552/4885NCF1 1129/4885BACE1 2807/4885
US-20130082209-A1 METAL COMPLEXES MCOLN2, MCOLN1, AP1M1 HTR3A 4398/4885NCF1 458/4885BACE1 1595/4885
US-20170309832-A1 METAL COMPLEXES SOD1, AP1M1, AP3M1 HTR3A 4552/4885NCF1 1129/4885BACE1 2807/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.