SCHEMBL13709258

SCHEMBL13709258

O=NCc1ccc2c(c1)N(c1ccccc1)CCC2

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.46
OPRM1 P35372 5/20 0.39
OPRK1 P41145 4/20 0.38
OPRD1 P41143 3/20 0.38
ALDH1A1 P00352 3/20 0.37
TP53 P04637 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.34
MGLL Q99685 1/20 0.34
MAPT P10636 1/20 0.34
RORC P51449 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
DRD2 P14416 1/20 0.34
DRD4 P21917 1/20 0.34
DRD3 P35462 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17275642 0.85 ACHE (0.48) ACHEOPRM1OPRK1OPRD1ALDH1A1
SCHEMBL3501876 0.82 ACHE (0.48) ACHEOPRM1OPRK1OPRD1SMN1; SMN2
SCHEMBL17276366 0.79 ACHE (0.43) ACHEOPRM1OPRK1OPRD1ALDH1A1
SCHEMBL17276390 0.79 ACHE (0.46) ACHEOPRM1OPRK1OPRD1
SCHEMBL2096904 0.77 DRD1 (0.48) ACHESMN1; SMN2MAPTCHRM2CHRM4
SCHEMBL25177736 0.75 BRD4 (0.48) ACHEALDH1A1TP53SMN1; SMN2MGLL
SCHEMBL3503283 0.74 ALDH1A1 (0.50) ACHEOPRM1ALDH1A1TP53SMN1; SMN2
SCHEMBL30317408 0.74 ROCK1 (0.48) ACHEALDH1A1SMN1; SMN2MAPT
SCHEMBL25184947 0.74 ROCK1 (0.48) ACHEALDH1A1SMN1; SMN2MAPT
SCHEMBL26149606 0.74 ACHE (0.43) ACHEOPRM1ALDH1A1TP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2096109-A1 CARBOXYLIC ACID DERIVATIVE Astellas Pharma Inc. (JP) 2009-09-02 EP disclosed