SCHEMBL13717048

SCHEMBL13717048

Cc1ccc(OC(N)(N)N)c(O)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.46
ALDH1A1 P00352 4/20 0.42
ALOX15 P16050 2/20 0.42
HSD17B10 Q99714 2/20 0.42
TP53 P04637 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
LMNA P02545 2/20 0.39
CYP3A4 P08684 1/20 0.39
CHRM1 P11229 1/20 0.39
SLC6A2 P23975 1/20 0.39
ADRA1A P35348 1/20 0.39
HTR2B P41595 1/20 0.39
AR P10275 1/20 0.39
ACHE P22303 2/20 0.39
GAA P10253 2/20 0.36
MAPT P10636 2/20 0.36
KMT2A Q03164 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14553749 0.80 TRPA1 (0.46) TRPA1ALDH1A1ALOX15HSD17B10TP53
SCHEMBL13463122 0.79 ALDH1A1 (0.42) ALDH1A1ALOX15TP53TDP1CA1
SCHEMBL10292484 0.76 TRPA1 (0.56) TRPA1ALDH1A1ALOX15HSD17B10TP53
SCHEMBL806486 0.76 ALDH1A1 (0.36) ALDH1A1CA1CA2CA9LMNA
SCHEMBL6441756 0.76 AR (0.43) TRPA1ALDH1A1ALOX15HSD17B10TP53
SCHEMBL6442340 0.76 ALDH1A1 (0.43) TRPA1ALDH1A1ALOX15HSD17B10TP53
SCHEMBL29398758 0.74 ACHE (0.62) TRPA1ALDH1A1ALOX15TP53TDP1
SCHEMBL218637 0.74 ACHE (0.62) TRPA1ALDH1A1ALOX15TP53TDP1
SCHEMBL13971412 0.72 TRPA1 (0.52) TRPA1ALDH1A1ALOX15HSD17B10TP53
SCHEMBL3371911 0.71 TRPA1 (0.45) TRPA1ALDH1A1ALOX15HSD17B10TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1427415-B1 LACTAM-CONTAINING COMPOUNDS AND DERIVATIVES THEREOF AS FACTOR XA INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2009-08-12 EP disclosed