SCHEMBL13728481

SCHEMBL13728481

COc1cncc2cc(F)ccc12

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 4/20 0.43
PDGFRB P09619 2/20 0.43
PDGFRA P16234 2/20 0.43
BRAF P15056 2/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
SCN9A Q15858 1/20 0.41
TDO2 P48775 2/20 0.39
TRPA1 O75762 2/20 0.39
IDO1 P14902 1/20 0.39
KCNH2 Q12809 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26317676 0.86 PDE10A (0.43) PDE10APDGFRBPDGFRABRAFCYP11B1
SCHEMBL30517018 0.79 POLB (0.40) PDE10ACYP11B1CYP11B2TDO2IDO1
SCHEMBL25840214 0.79 POLB (0.40) PDE10ACYP11B1CYP11B2TDO2IDO1
SCHEMBL27983652 0.79 PDE10A (0.43) PDE10ACYP11B1CYP11B2
SCHEMBL13729147 0.76 PDE10A (0.38) PDE10APDGFRBPDGFRATRPA1
SCHEMBL24773765 0.76 ACHE (0.53) PDGFRBPDGFRATRPA1
SCHEMBL1536378 0.73 CYP11B1 (0.49) PDE10ABRAFCYP11B1CYP11B2
SCHEMBL22559289 0.72 LCK (0.50) PDE10ACYP11B1CYP11B2
SCHEMBL20975068 0.72 CYP11B2 (0.37) BRAFCYP11B1CYP11B2TDO2IDO1
SCHEMBL30701983 0.72 CYP11B2 (0.37) BRAFCYP11B1CYP11B2TDO2IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2909205-A1 HEPATITIS C VIRUS INHIBITORS Bristol-Myers Squibb Company (US) 2015-08-26 EP disclosed
WO-2014062196-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2014-04-24 WO disclosed
EP-2705049-A1 HEPATITIS C VIRUS INHIBITORS Bristol-Myers Squibb Company (US) 2014-03-12 EP disclosed
WO-2012151195-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-11-08 WO disclosed