SCHEMBL13729601

SCHEMBL13729601

O=C(NCc1cccc(Oc2ccccc2)c1)c1ccncn1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 2/20 0.56
MMP13 P45452 4/20 0.54
CYP3A4 P08684 4/20 0.54
MAPK14 Q16539 3/20 0.54
LMNA P02545 1/20 0.54
HTT P42858 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
CCR8 P51685 1/20 0.53
KCNH2 Q12809 1/20 0.53
ROCK2 O75116 4/20 0.51
ROCK1 Q13464 4/20 0.49
CYP2D6 P10635 3/20 0.49
CYP2C9 P11712 3/20 0.49
MAPK8 P45983 1/20 0.49
PRKACA P17612 2/20 0.48
PRKX P51817 2/20 0.48
PRKCQ Q04759 2/20 0.48
GRK5 P34947 1/20 0.48
GSK3A P49840 1/20 0.48
GSK3B P49841 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5252907 0.87 ROCK2 (0.64) MMP13CYP3A4LMNAHTTSMN1; SMN2
SCHEMBL27965276 0.85 MMP13 (0.69) MMP13HTTSMN1; SMN2ROCK2ROCK1
SCHEMBL27931805 0.84 ROCK2 (0.66) MMP13MAPK14ROCK2ROCK1
SCHEMBL13729131 0.80 MMP13 (0.52) MMP13HTTSMN1; SMN2CYP2C9HPGD
SCHEMBL13728776 0.80 CCR8 (0.55) MMP13CYP3A4MAPK14LMNAHTT
Tert-Butylamine SCHEMBL28093817 0.79 ROCK2 (0.60) MMP13MAPK14ROCK2ROCK1
SCHEMBL13728282 0.79 ROCK2 (0.55) MMP13CYP3A4HTTSMN1; SMN2ROCK2
SCHEMBL13729455 0.78 MAPK14 (0.50) MMP13CYP3A4MAPK14LMNAHTT
SCHEMBL1681517 0.77 POLB (0.53) FFAR1MMP13MAPK14LMNAMAPK8
SCHEMBL28042144 0.77 MAPK8 (0.51) FFAR1MMP13CYP3A4MAPK14LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012151567-A1 PYRIMIDINONE COMPOUNDS AND METHODS FOR PREVENTING AND TREATING INFLUENZA ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 2012-11-08 WO disclosed