Gentisic Acid

Gentisic Acid

SCHEMBL13729892

CC(N)CCc1cc(F)c(F)cc1F.O=C(O)c1cc(O)ccc1O

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.49
CA2 P00918 4/20 0.49
CA12 O43570 3/20 0.49
CA7 P43166 3/20 0.49
CA9 Q16790 3/20 0.49
CA14 Q9ULX7 3/20 0.49
PTGS2 P35354 2/20 0.49
ALOX5 P09917 1/20 0.49
CHRNA7 P36544 1/20 0.46
LCK P06239 5/20 0.44
EGFR P00533 3/20 0.44
ALDH1A1 P00352 6/20 0.40
TDP1 Q9NUW8 5/20 0.40
TYR P14679 2/20 0.40
MAPT P10636 2/20 0.40
RGS12 O14924 1/20 0.40
CAMKK2 Q96RR4 1/20 0.40
NOX4 Q9NPH5 1/20 0.40
HPGD P15428 5/20 0.39
MEN1 O00255 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Gentisic Acid SCHEMBL13732886 0.81 CA12 (0.49) CA1CA2CA12CA7CA9
SCHEMBL4697922 0.77 DPP4 (0.55)
SCHEMBL13729895 0.76 CA12 (0.46) CA1CA2CA12CA7CA9
Trifluoroacetic Acid SCHEMBL3134971 0.76 DPP4 (0.42) CYP3A4
Adipic Acid SCHEMBL13729711 0.75 GABRP (0.44) ALDH1A1
Hydrochloric Acid SCHEMBL13730064 0.75 DPP4 (0.53)
Phosphoric Acid SCHEMBL13730179 0.74 DPP4 (0.46) ALDH1A1TDP1CYP3A4
Phosphoric Acid SCHEMBL14128619 0.73 DPP4 (0.45) ALDH1A1TDP1CYP3A4
Gentisic Acid SCHEMBL28318579 0.70 CA1 (0.91) CA1CA2CA12CA7CA9
Gentisic Acid SCHEMBL29349919 0.70 CA1 (1.00) CA1CA2CA12CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2681220-A2 NOVEL SALTS OF DPP-IV INHIBITOR Cadila Healthcare Limited (IN) 2014-01-08 EP claimed
WO-2012147092-A2 NOVEL SALTS OF DPP-IV INHIBITOR CADILA HEALTHCARE LIMITED (IN) 2012-11-01 WO claimed
EP-2681220-A2 NOVEL SALTS OF DPP-IV INHIBITOR Cadila Healthcare Limited (IN) 2014-01-08 EP disclosed
WO-2012147092-A2 NOVEL SALTS OF DPP-IV INHIBITOR CADILA HEALTHCARE LIMITED (IN) 2012-11-01 WO disclosed