SCHEMBL13737906

SCHEMBL13737906

O=C(O)N1CC=Cc2ccccc2C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.44
NAMPT P43490 8/20 0.40
HSD17B3 P37058 1/20 0.39
TAS1R3 Q7RTX0 1/20 0.38
TAS1R1 Q7RTX1 1/20 0.38
TAS1R2 Q8TE23 1/20 0.38
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38
HSP90B1 P14625 1/20 0.38
TRAP1 Q12931 1/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
HDAC8 Q9BY41 2/20 0.37
NPC1 O15118 1/20 0.37
TP53 P04637 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
RYR2 Q92736 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25252621 0.77 DPP9 (0.40) NAMPTTAS1R3TAS1R1TAS1R2HSP90B1
SCHEMBL2533362 0.76 NOTUM (0.64) NOTUMNAMPTTAS1R3TAS1R1TAS1R2
SCHEMBL29758685 0.76 NOTUM (0.64) NOTUMNAMPTTAS1R3TAS1R1TAS1R2
SCHEMBL304994 0.73 HDAC3 (0.43) NOTUMNAMPTHSD17B3TAS1R3TAS1R1
SCHEMBL29950507 0.73 HDAC3 (0.43) NOTUMNAMPTHSD17B3TAS1R3TAS1R1
SCHEMBL15323808 0.72 HSD17B3 (0.40) NOTUMNAMPTHSD17B3TAS1R3TAS1R1
SCHEMBL13236581 0.72 MAOA (0.45) HSD17B3MEN1MAPTKMT2ATP53
Hydrochloric Acid SCHEMBL7007436 0.71 HDAC3 (0.43) NOTUMNAMPTHSD17B3TAS1R3TAS1R1
Indene SCHEMBL30959780 0.71 CA2 (0.47) NOTUMHSD17B3MAPT
Indene SCHEMBL6700608 0.71 CA2 (0.47) NOTUMHSD17B3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2707358-A1 BENZAZEPINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, AND THEIR USE IN THERAPY Abbvie Deutschland GmbH & Co. KG (DE) 2014-03-19 EP disclosed
WO-2012152915-A1 BENZAZEPINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, AND THEIR USE IN THERAPY ABBOTT GMBH & CO. KG (DE) 2012-11-15 WO disclosed