SCHEMBL13745966

SCHEMBL13745966

Cc1nc([C@H]2C[C@@H]3[C@H](C2)C3(F)F)c(-c2ccc(Cl)nc2)c(=O)[nH]1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TYMS P04818 3/20 0.32
PIK3CA P42336 2/20 0.32
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
NPC1 O15118 2/20 0.31
RAB9A P51151 1/20 0.31
HPGD P15428 1/20 0.30
HTT P42858 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13746006 0.87 TYMS (0.39) TYMSKDM4EALDH1A1HPGDHTT
SCHEMBL13746627 0.84 USP1 (0.34) TYMSPIK3CAKDM4EALDH1A1NPC1
SCHEMBL13746667 0.81 PDE2A (0.37) TYMSPIK3CA
SCHEMBL13746623 0.77 FASN (0.37)
SCHEMBL13746305 0.72 TYMS (0.41) TYMSKDM4EHPGDHTT
SCHEMBL13746236 0.72 TYMS (0.41) TYMSKDM4EHPGDHTT
SCHEMBL13746410 0.71 TYMS (0.39) TYMSKDM4EALDH1A1HPGD
SCHEMBL4755648 0.68 PIK3CA (0.35) PIK3CA
SCHEMBL13746295 0.68
SCHEMBL13745968 0.68 PIK3CA (0.36) TYMSPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100403-A1 SUBSTITUTED ARYL PYRIMIDINONES NEUROGEN CORPORATION (US) 2009-08-13 WO disclosed