SCHEMBL4755648

SCHEMBL4755648

Cc1nc(C2CC3C(C2)C3(F)F)[nH]c(=O)c1-c1ccc(C#N)nc1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.35
KDM5B Q9UGL1 1/20 0.34
VHL P40337 1/20 0.32
DGAT1 O75907 1/20 0.32
PDE4A P27815 2/20 0.32
SYK P43405 1/20 0.32
ALOX5AP P20292 1/20 0.31
PDE9A O76083 2/20 0.31
MAPK1 P28482 1/20 0.30
KDM1A O60341 1/20 0.30
SCN10A Q9Y5Y9 1/20 0.30
KRAS P01116 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4753259 0.82 PIK3CA (0.35) PIK3CAKDM5BVHLDGAT1PDE4A
SCHEMBL4753738 0.77 JAK2 (0.35) PIK3CAKDM5BVHLDGAT1PDE4A
SCHEMBL4753279 0.72 FASN (0.32) PDE9A
SCHEMBL4753233 0.71 PDE9A (0.37) PDE9AKDM1A
SCHEMBL13745966 0.68 TYMS (0.32) PIK3CA
SCHEMBL13985419 0.68 PDE4B (0.34) PIK3CASYKKDM1A
SCHEMBL4756614 0.67 KDM4E (0.33)
SCHEMBL13746012 0.67 PIK3CA (0.36) PIK3CAKDM5BVHLDGAT1PDE4A
SCHEMBL4756695 0.65 HSD11B1 (0.39) PDE9AKDM1A
SCHEMBL13660413 0.62 DPP4 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008156607-A1 SUBSTITUTED PYRIMIDINONES NEUROGEN CORPORATION (US) 2008-12-24 WO claimed
WO-2008156607-A1 SUBSTITUTED PYRIMIDINONES NEUROGEN CORPORATION (US) 2008-12-24 WO disclosed