SCHEMBL13745968

SCHEMBL13745968

CNc1nc([C@H]2CC[C@@H](C(F)(F)F)CC2)c(-c2ccc(Cl)nc2)c(=O)[nH]1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.36
PI4KB Q9UBF8 1/20 0.33
TYMS P04818 1/20 0.33
JAK2 O60674 1/20 0.31
JAK1 P23458 1/20 0.31
TYK2 P29597 1/20 0.31
EIF4E P06730 1/20 0.31
SPR P35270 1/20 0.31
RPS6KB1 P23443 1/20 0.31
GRIA1 P42261 2/20 0.30
PDE2A O00408 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13746941 0.88 EIF4E (0.36) TYMSJAK2JAK1TYK2EIF4E
SCHEMBL13746667 0.87 PDE2A (0.37) PIK3CAPI4KBTYMSJAK2JAK1
SCHEMBL13746668 0.82 TYMS (0.36) TYMSJAK2JAK1TYK2PDE2A
SCHEMBL13746627 0.78 USP1 (0.34) PIK3CATYMSSPRRPS6KB1PDE2A
SCHEMBL4020404 0.76 PDE2A (0.49) PIK3CAPI4KBGRIA1PDE2A
SCHEMBL4023129 0.75 PDE2A (0.37) PI4KBTYMSJAK2JAK1TYK2
SCHEMBL4023133 0.75 PDE2A (0.37) PI4KBTYMSJAK2JAK1TYK2
SCHEMBL13747129 0.73 TYMS (0.38) TYMSPDE2A
SCHEMBL13746960 0.72 TYMS (0.39) TYMS
SCHEMBL13746012 0.72 PIK3CA (0.36) PIK3CAPI4KBJAK2JAK1TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100403-A1 SUBSTITUTED ARYL PYRIMIDINONES NEUROGEN CORPORATION (US) 2009-08-13 WO disclosed