SCHEMBL13748544

SCHEMBL13748544

Cc1cc(-n2cc3c(n2)CCN(CC(=O)N2CCC(N4CCCC4)C2)C3)ccn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 9/20 0.42
KCNH2 Q12809 4/20 0.38
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
POLB P06746 2/20 0.35
CHRM4 P08173 1/20 0.35
GAA P10253 1/20 0.35
TSHR P16473 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
G6PD P11413 1/20 0.35
HPGD P15428 1/20 0.35
CACNA1B Q00975 1/20 0.35
APBA1 Q02410 1/20 0.35
HSD17B10 Q99714 1/20 0.35
APOBEC3G Q9HC16 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
PRMT5 O14744 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13748066 0.95 SLC6A9 (0.43) SLC6A9KCNH2CYP2D6CYP2C19NPSR1
SCHEMBL13748637 0.94 SLC6A9 (0.43) SLC6A9KCNH2CYP2D6CYP2C19NPSR1
SCHEMBL13748776 0.94 SLC6A9 (0.43) SLC6A9KCNH2CYP2D6CYP2C19NPSR1
SCHEMBL13748663 0.88 KDM4E (0.44) SLC6A9KCNH2KDM4EALDH1A1PRMT5
SCHEMBL13749074 0.88 SLC6A9 (0.42) SLC6A9KCNH2CYP2D6CYP2C19NPSR1
SCHEMBL13748854 0.88 SLC6A9 (0.43) SLC6A9KCNH2NPSR1CHRM4KDM4E
SCHEMBL4067642 0.88 SLC6A9 (0.43) SLC6A9KCNH2NPSR1KDM4EALDH1A1
SCHEMBL13749102 0.86 SLC6A9 (0.43) SLC6A9KCNH2CHRM4
SCHEMBL13749138 0.85 SLC6A9 (0.43) SLC6A9KCNH2CHRM4KDM4EALDH1A1
SCHEMBL13748690 0.84 SLC6A9 (0.42) SLC6A9KCNH2CHRM4PRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100120-A2 PYRIDINYL-SUBSTITUTED PIPERAZINYL OXOETHYL TETRAHYDROPYRAZOLOPYRIDINES NEUROGEN CORPORATION (US) 2009-08-13 WO disclosed