SCHEMBL13748637

SCHEMBL13748637

Cc1cc(-n2cc3c(n2)CCN(CC(=O)N2CCC(N4CCCCCC4)CC2)C3)ccn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 9/20 0.43
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
TSHR P16473 1/20 0.40
MAPT P10636 1/20 0.40
G6PD P11413 1/20 0.40
HPGD P15428 1/20 0.40
CACNA1B Q00975 1/20 0.40
APBA1 Q02410 1/20 0.40
HSD17B10 Q99714 1/20 0.40
APOBEC3G Q9HC16 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
KCNH2 Q12809 4/20 0.38
IRAK4 Q9NWZ3 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13748776 1.00 SLC6A9 (0.43) SLC6A9CYP2D6CYP2C19NPSR1KDM4E
SCHEMBL13748066 0.99 SLC6A9 (0.43) SLC6A9CYP2D6CYP2C19NPSR1KDM4E
SCHEMBL13748544 0.94 SLC6A9 (0.42) SLC6A9CYP2D6CYP2C19NPSR1KDM4E
SCHEMBL13748663 0.92 KDM4E (0.44) SLC6A9KDM4EALDH1A1KCNH2IRAK4
SCHEMBL13749074 0.92 SLC6A9 (0.42) SLC6A9CYP2D6CYP2C19NPSR1KDM4E
SCHEMBL4067642 0.92 SLC6A9 (0.43) SLC6A9NPSR1KDM4EALDH1A1KCNH2
SCHEMBL13748854 0.92 SLC6A9 (0.43) SLC6A9NPSR1KDM4EALDH1A1KCNH2
SCHEMBL13748980 0.87 SLC6A9 (0.41) SLC6A9KDM4EALDH1A1TSHRMAPT
SCHEMBL13748801 0.86 SLC6A9 (0.41) SLC6A9KDM4EALDH1A1TSHRMAPT
SCHEMBL13748936 0.85 SLC6A9 (0.40) SLC6A9KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100120-A2 PYRIDINYL-SUBSTITUTED PIPERAZINYL OXOETHYL TETRAHYDROPYRAZOLOPYRIDINES NEUROGEN CORPORATION (US) 2009-08-13 WO disclosed