SCHEMBL13754686

SCHEMBL13754686

Cc1[nH]c(C)c(-c2ccc(OCc3ccccc3)nc2)c(=O)c1Cl

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.56
LOXL2 Q9Y4K0 1/20 0.43
BRD4 O60885 4/20 0.42
CREBBP Q92793 1/20 0.42
PKM P14618 1/20 0.42
POLB P06746 1/20 0.40
IKBKE Q14164 1/20 0.38
FFAR1 O14842 4/20 0.38
GABRP O00591 1/20 0.38
GABRD O14764 1/20 0.38
GABRA1 P14867 1/20 0.38
GABRB1 P18505 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38
GABRA2 P47869 1/20 0.38
GABRB2 P47870 1/20 0.38
GABRA4 P48169 1/20 0.38
GABRE P78334 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4469233 0.89 SLC2A1 (0.52) SLC2A1LOXL2BRD4CREBBPGABRA5
SCHEMBL13754685 0.86 SLC2A1 (0.73) SLC2A1LOXL2BRD4CREBBPPKM
SCHEMBL4490726 0.86 SLC2A1 (0.61) SLC2A1GABRA5
SCHEMBL4484452 0.85 SLC2A1 (0.53) SLC2A1
SCHEMBL4468888 0.85 SLC2A1 (0.79) SLC2A1
SCHEMBL4476493 0.84 SLC2A1 (0.52) SLC2A1
SCHEMBL4476932 0.83 GPR84 (0.48) SLC2A1MAT2AMCL1
SCHEMBL4487955 0.83 SLC2A1 (0.66) SLC2A1
SCHEMBL4493447 0.82 SLC2A1 (0.52) SLC2A1FFAR1
SCHEMBL3397585 0.81 SLC2A1 (0.43) SLC2A1BRD4CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7579353-B2 Pyridinone derivatives against malaria GLAXO GROUP LIMITED (GB) 2009-08-25 US disclosed
US-20080287461-A1 Pyridinone Derivatives Against Malaria GLAXO GROUP LIMITED (GB) 2008-11-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080287461-A1 Pyridinone Derivatives Against Malaria G6PD, PNPO, PLPBP SLC2A1 2278/4885LOXL2 2417/4885BRD4 2655/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.