SCHEMBL1375993

SCHEMBL1375993

c1nc2nc(C3CCC3)ncc2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAK1 Q13153 2/20 0.51
ALDH1A1 P00352 1/20 0.49
KDM4E B2RXH2 1/20 0.49
CDK2 P24941 3/20 0.40
RXFP1 Q9HBX9 1/20 0.40
ALOX5AP P20292 2/20 0.36
FEN1 P39748 2/20 0.36
SCD O00767 2/20 0.35
CCNT1 O60563 1/20 0.34
CDK1 P06493 1/20 0.34
CCNB1 P14635 1/20 0.34
CDK7 P50613 1/20 0.34
CDK9 P50750 1/20 0.34
CCNH P51946 1/20 0.34
ADORA1 P30542 1/20 0.34
HTR2B P41595 1/20 0.34
POLA1 P09884 1/20 0.33
CCNE1 P24864 1/20 0.32
CDK5 Q00535 1/20 0.32
KDM5B Q9UGL1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2951841 0.97 PAK1 (0.55) PAK1ALDH1A1KDM4ECDK2RXFP1
SCHEMBL10869151 0.95 PAK1 (0.57) PAK1ALDH1A1KDM4ECDK2RXFP1
Hydrochloric Acid SCHEMBL6821631 0.95 PAK1 (0.54) PAK1ALDH1A1KDM4ECDK2RXFP1
SCHEMBL31380702 0.85 ALDH1A1 (0.45) PAK1ALDH1A1KDM4ECDK2RXFP1
SCHEMBL4373728 0.81 ALDH1A1 (0.44) PAK1ALDH1A1KDM4ECDK2RXFP1
SCHEMBL9854792 0.77 ALDH1A1 (0.46) PAK1ALDH1A1KDM4ECDK2RXFP1
SCHEMBL2388908 0.76 PAK1 (0.46) PAK1ALDH1A1KDM4ECDK2RXFP1
SCHEMBL5872330 0.75 PAK1 (0.45) PAK1ALDH1A1KDM4ECDK2RXFP1
SCHEMBL2002538 0.75 PAK1 (0.48) PAK1ALDH1A1KDM4ECDK2RXFP1
SCHEMBL2953152 0.75 ALDH1A1 (0.45) PAK1ALDH1A1KDM4ECDK2RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106305279-A Comprehensive management and cultivation method for promoting rapid propagation of poplar seedlings 梁国婷 2017-01-11 CN claimed
US-9273050-B2 Cyclobutyl purine derivative, angiogenesis promoting agent, lumen formation promoting agent, neurocyte growth promoting agent, and drug NATIONAL UNIVERSITY CORPORATION KAGAWA UNIVERSITY (JP) 2016-03-01 US claimed
EP-2377865-B1 CYCLOBUTYL PURINE DERIVATIVE, ANGIOGENESIS PROMOTING AGENT, LUMENIZATION PROMOTING AGENT, NEUROCYTE GROWTH PROMOTING AGENT, AND DRUG UNIV KAGAWA NAT UNIV CORP (JP) 2014-12-17 EP claimed
CN-102227427-B Cyclobutyl purine derivative, angiogenesis promoting agent, lumenization promoting agent, neurocyte growth promoting agent, and drug UNIV KAGAWA NAT UNIV CORP (JP) 2014-04-02 CN claimed
CN-102227427-A Cyclobutyl purine derivative, angiogenesis promoting agent, lumenization promoting agent, neurocyte growth promoting agent, and drug UNIV KAGAWA NAT UNIV CORP (JP) 2011-10-26 CN claimed
EP-2377865-A1 CYCLOBUTYL PURINE DERIVATIVE, ANGIOGENESIS PROMOTING AGENT, LUMENIZATION PROMOTING AGENT, NEUROCYTE GROWTH PROMOTING AGENT, AND DRUG National University Corporation Kagawa University (JP) 2011-10-19 EP claimed
US-20110230659-A1 CYCLOBUTYL PURINE DERIVATIVE, ANGIOGENESIS PROMOTING AGENT, LUMEN FORMATION PROMOTING AGENT, NEUROCYTE GROWTH PROMOTING AGENT, AND DRUG NATIONAL UNIVERSITY CORPORATION KAGAWA UNIVERSITY (JP) 2011-09-22 US claimed
US-5874578-A Process for preparing guanine-containing antiviral agents and purinyl salts useful in such process BRISTOL-MYERS SQUIBB (US) 1999-02-23 US claimed
CN-1036712-C Process for preparing guanine-containing antiviral agents and purinyl salts useful in such process SQUIBB & SONS INC (US) 1997-12-17 CN claimed
CN-1083813-A Contain guanine antiviral agent the preparation method and be used for the purine salt of this method SQUIBB & SONS INC (US) 1994-03-16 CN claimed
EP-0579421-A2 Process for preparing guanine-containing antiviral agents and purinyl salts useful in such process E.R. Squibb & Sons, Inc. (US) 1994-01-19 EP claimed
US-12202850-B2 Cyclobutyl purine derivative or salt thereof FUJIFILM CORPORATION (JP) 2025-01-21 US disclosed
US-12202850-B2 Cyclobutyl purine derivative or salt thereof FUJIFILM CORPORATION (JP) 2025-01-21 US disclosed
US-20230295202-A1 CYCLOBUTYL PURINE DERIVATIVE OR SALT THEREOF FUJIFILM CORPORATION (JP) 2023-09-21 US disclosed
US-20230295202-A1 CYCLOBUTYL PURINE DERIVATIVE OR SALT THEREOF FUJIFILM CORPORATION (JP) 2023-09-21 US disclosed
EP-0579421-A2 Process for preparing guanine-containing antiviral agents and purinyl salts useful in such process E.R. Squibb & Sons, Inc. (US) 1994-01-19 EP disclosed
EP-0554025-A2 Fluorinated cyclobutyl purines and pyrimidines E.R. SQUIBB & SONS, INC. (US) 1993-08-04 EP disclosed
WO-1991018969-A1 FLUORINATED BIS(HYDROXYMETHYL)CYCLOBUTYL PURINES AND PYRIMIDINES E.R. SQUIBB & SONS, INC. (US) 1991-12-12 WO disclosed
CN-1036575-A The method of two (methylol) cyclobutyl purine of preparation and pyrimidine SQUIBB & SONS INC (US) 1989-10-25 CN disclosed
CN-1036575-A The method of two (methylol) cyclobutyl purine of preparation and pyrimidine SQUIBB & SONS INC (US) 1989-10-25 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230295202-A1 CYCLOBUTYL PURINE DERIVATIVE OR SALT THEREOF SLC28A1, SLC20A1, SLC29A1 PAK1 2882/4885ALDH1A1 504/4885KDM4E 4331/4885
US-20110230659-A1 CYCLOBUTYL PURINE DERIVATIVE, ANGIOGENESIS PROMOTING AGENT, LUMEN FORMATION PROMOTING AGENT, NEUROCYTE GROWTH PROMOTING AGENT, AND DRUG DCX, MKI67, SLC29A1 PAK1 2235/4885ALDH1A1 1340/4885KDM4E 4808/4885
US-12202850-B2 Cyclobutyl purine derivative or salt thereof SLC28A1, SLC20A1, SLC29A1 PAK1 2882/4885ALDH1A1 504/4885KDM4E 4331/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.