SCHEMBL4373728

SCHEMBL4373728

c1nc2nc(C3CCNC3)ncc2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
KDM4E B2RXH2 1/20 0.44
PAK1 Q13153 1/20 0.43
CDK2 P24941 2/20 0.36
RXFP1 Q9HBX9 1/20 0.36
HRH3 Q9Y5N1 4/20 0.36
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
SCD O00767 2/20 0.33
HTR3A P46098 1/20 0.33
HRH4 Q9H3N8 3/20 0.32
CCNT1 O60563 1/20 0.32
CDK1 P06493 1/20 0.32
CCNB1 P14635 1/20 0.32
CDK7 P50613 1/20 0.32
CDK9 P50750 1/20 0.32
CCNH P51946 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1375993 0.81 PAK1 (0.51) ALDH1A1KDM4EPAK1CDK2RXFP1
SCHEMBL2951841 0.81 PAK1 (0.55) ALDH1A1KDM4EPAK1CDK2RXFP1
SCHEMBL10869151 0.80 PAK1 (0.57) ALDH1A1KDM4EPAK1CDK2RXFP1
Hydrochloric Acid SCHEMBL6821631 0.80 PAK1 (0.54) ALDH1A1KDM4EPAK1CDK2RXFP1
SCHEMBL31380702 0.77 ALDH1A1 (0.45) ALDH1A1KDM4EPAK1CDK2RXFP1
SCHEMBL4373719 0.76 HRH3 (0.36) HRH3CHRNB2CHRNA4HTR3AHRH4
SCHEMBL18167360 0.75 ALDH1A1 (0.41) ALDH1A1KDM4EPAK1
SCHEMBL9854792 0.72 ALDH1A1 (0.46) ALDH1A1KDM4EPAK1CDK2RXFP1
SCHEMBL12539876 0.71 TYRO3 (0.46) SCDCDK7CDK9
SCHEMBL1378385 0.70 ALDH1A1 (0.47) ALDH1A1KDM4EPAK1CDK2RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1113020-B1 Nucleosides and oligonucleotides containing boron clusters UNIV EMORY (US) 2009-10-28 EP disclosed
US-6583122-B2 Use in boron neutron capture therapy (BNCT) and diagnostic purposes; treating cancer, viral infections such as HIV, hepatitis B virus EMORY UNIVERSITY 2003-06-24 US disclosed
US-20020160969-A1 Nucleosides and oligonucleotides containing boron clusters DEPARTMENT OF VETERANS AFFAIRS 2002-10-31 US disclosed
EP-0731808-B1 NUCLEOSIDES AND OLIGONUCLEOTIDES CONTAINING BORON CLUSTERS UNIV EMORY (US) 2001-07-11 EP disclosed
EP-1113020-A2 Nucleosides and oligonucleotides containing boron clusters EMORY UNIVERSITY (US) 2001-07-04 EP disclosed
US-6180766-B1 OLIGONUCLEOTIDE WITH UNCHARGED INTERNUCLEOTIDE LINKAGE(S) OF 3',5'-O,O-((CARBORAN-1-YL-METHYL)PHOSPHONATE); MADE BY REACTING O-METHYL(O-CARBORAN-1-YL)METHYL PHOSPHONATE WITH PROTECTED NUCLEOSIDE; USE IN BORON NEUTRON CAPTURE THERAPY DEPARTMENT OF VETERANS AFFAIRS 2001-01-30 US disclosed
US-5872107-A ANTICARCINOGENIC AGENTS CAPTURE THERAPY FOR TUMORS EMORY UNIVERSITY (US) 1999-02-16 US disclosed
EP-0788364-A4 TREATMENT OF UROGENITAL CANCER WITH BORON NEUTRON CAPTURE THERAPY UNIV EMORY (US) 1998-05-06 EP disclosed
EP-0788364-A1 TREATMENT OF UROGENITAL CANCER WITH BORON NEUTRON CAPTURE THERAPY EMORY UNIVERSITY (US) 1997-08-13 EP disclosed
EP-0731808-A4 NUCLEOSIDES AND OLIGONUCLEOTIDES CONTAINING BORON CLUSTERS UNIV EMORY (US) 1997-04-02 EP disclosed
US-5599796-A USING BORON CLUSTER-CONTAINING NUCLEOSIDES OR OLIGONUCLEOTIDES; PARTICULARLY EFFECTIVE FOR BLADDER, PROSTATE AND KIDNEY EMORY UNIVERSITY (US) 1997-02-04 US disclosed
EP-0731808-A1 NUCLEOSIDES AND OLIGONUCLEOTIDES CONTAINING BORON CLUSTERS EMORY UNIVERSITY (US) 1996-09-18 EP disclosed
WO-1996014073-A1 TREATMENT OF UROGENITAL CANCER WITH BORON NEUTRON CAPTURE THERAPY EMORY UNIVERSITY (US) 1996-05-17 WO disclosed
WO-1995015333-A1 NUCLEOSIDES AND OLIGONUCLEOTIDES CONTAINING BORON CLUSTERS EMORY UNIVERSITY (US) 1995-06-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020160969-A1 Nucleosides and oligonucleotides containing boron clusters NUDT1, NTPCR, NAMPT ALDH1A1 4697/4885KDM4E 4815/4885PAK1 4433/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.