SCHEMBL13763542

SCHEMBL13763542

CCc1ccc(NCCN2CCCC2)nc1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.58
CYP1A2 P05177 1/20 0.57
CYP2D6 P10635 1/20 0.57
NMT1 P30419 1/20 0.49
HRH4 Q9H3N8 1/20 0.48
ACHE P22303 2/20 0.46
TLR7 Q9NYK1 2/20 0.45
SIGMAR1 Q99720 6/20 0.44
TRPC5 Q9UL62 1/20 0.44
MAP3K11 Q16584 1/20 0.42
KCNH2 Q12809 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2056410 0.87 KDR (0.48) CYP1A2CYP2D6SIGMAR1TRPC5
SCHEMBL1108663 0.82 NMT1 (0.54) HRH3NMT1HRH4ACHETLR7
SCHEMBL14924463 0.81 NMT1 (0.56) HRH3NMT1HRH4ACHETLR7
SCHEMBL21412819 0.80 DPP7 (0.48) HRH3CYP1A2CYP2D6NMT1HRH4
SCHEMBL2320244 0.79 NMT1 (0.51) HRH3NMT1HRH4ACHESIGMAR1
SCHEMBL4069152 0.79 HRH3 (0.62) HRH3NMT1HRH4ACHETLR7
SCHEMBL2998111 0.79 NMT1 (0.48) HRH3CYP1A2CYP2D6NMT1HRH4
SCHEMBL13757473 0.78 NMT1 (0.48) HRH3NMT1HRH4ACHESIGMAR1
SCHEMBL15247195 0.78 NMT1 (0.48) HRH3NMT1HRH4ACHETLR7
SCHEMBL14238180 0.78 ALDH1A1 (0.51) HRH3NMT1HRH4ACHEMAP3K11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7579348-B2 Derivatives of 8-substituted xanthines PGXHEALTH, LLC (US) 2009-08-25 US disclosed
US-20070249598-A1 Derivatives of 8-substituted xanthines ADENOSINE THERAPEUTICS, LLC 2007-10-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070249598-A1 Derivatives of 8-substituted xanthines ADORA2B, ADORA2A, ADORA3 HRH3 354/4885CYP1A2 262/4885CYP2D6 399/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.