SCHEMBL13764677

SCHEMBL13764677

CC(=O)N1CCC(Oc2ccc(Br)cc2C=O)CC1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 2/20 0.50
PTGDR2 Q9Y5Y4 1/20 0.45
PDE4B Q07343 1/20 0.44
ALK Q9UM73 1/20 0.42
CHUK O15111 1/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
RAB9A P51151 2/20 0.41
PLA2G1B P04054 1/20 0.40
ATG4B Q9Y4P1 1/20 0.40
KDM1A O60341 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
POLB P06746 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
EGFR P00533 1/20 0.39
KDR P35968 1/20 0.39
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL274655 0.85 PDE4B (0.52) PDE4BKDM1A
SCHEMBL18003630 0.81 POLB (0.49) PTGDR2PDE4BPLA2G1BATG4BPOLB
SCHEMBL3400187 0.81 PDE4B (0.49) PDE4BKDM1A
SCHEMBL279184 0.81 PDE4B (0.49) PDE4BKDM1A
SCHEMBL3400190 0.81 PDE4B (0.49) PDE4BKDM1A
SCHEMBL275132 0.76 PTGDR2 (0.44) PTGDR2PDE4BPLA2G1BATG4BPOLB
SCHEMBL13815410 0.76 IKBKB (0.48) IKBKBPDE4BCHUKKMT2AMEN1
SCHEMBL31370640 0.76 ALDH1A1 (0.55) IKBKBALKKMT2AMEN1KDM1A
SCHEMBL223707 0.75 GPR119 (0.45) IKBKBPDE4BCHUKKMT2AMEN1
SCHEMBL3688993 0.75 MAPT (0.52) KMT2AMEN1RAB9APOLBNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080488-A1 SPIROINDOLINONE DERIVATIVES AS ANTICANCER AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2009-07-02 WO disclosed