SCHEMBL13772811

SCHEMBL13772811

Bc1cc(CC)ccc1Br

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.41
CYP2A6 P11509 2/20 0.40
CYP1A2 P05177 1/20 0.40
MAPT P10636 3/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.35
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 1/20 0.35
LMNA P02545 1/20 0.35
MAPK1 P28482 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CA2 P00918 1/20 0.34
EDNRB P24530 2/20 0.34
EDNRA P25101 2/20 0.34
KIF11 P52732 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
TP53 P04637 1/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14565700 0.82 TRPA1 (0.41) TRPA1CYP2A6CYP1A2MAPTRAB9A
SCHEMBL14565787 0.78 TRPA1 (0.46) TRPA1CYP2A6CYP1A2MAPTRAB9A
SCHEMBL4798301 0.78 TRPA1 (0.46) TRPA1CYP2A6CYP1A2MAPTRAB9A
SCHEMBL13772758 0.74 TRPA1 (0.43) TRPA1CYP2A6CYP1A2MAPTRAB9A
SCHEMBL10871333 0.74 TRPA1 (0.43) TRPA1CYP2A6CYP1A2MAPTRAB9A
SCHEMBL11797035 0.74 TRPA1 (0.43) TRPA1CYP2A6CYP1A2MAPTRAB9A
SCHEMBL19676665 0.74 TRPA1 (0.39) TRPA1CYP2A6CYP1A2MAPTRAB9A
SCHEMBL10208289 0.73 TRPA1 (0.64) TRPA1CYP2A6CYP1A2MAPTRAB9A
SCHEMBL257061 0.73 ALDH1A1 (0.42) TRPA1CYP2A6CYP1A2MAPTRAB9A
SCHEMBL14899824 0.73 NOS3 (0.42) TRPA1CYP2A6CYP1A2MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732917-B1 SELECTED CGRP ANTAGONISTS, METHODS FOR THE PRODUCTION THEREOF AND THEIR USE AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA (DE) 2009-07-29 EP disclosed