SCHEMBL13788811

SCHEMBL13788811

Nc1nc(N)c2c(Cc3ccc([N+](=O)[O-])cc3)csc2n1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DHFR P00374 2/20 0.44
POLB P06746 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
MAPT P10636 1/20 0.40
GAA P10253 1/20 0.39
IDO1 P14902 2/20 0.39
GHSR Q92847 2/20 0.39
LOXL2 Q9Y4K0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13788810 0.82 PIK3CD (0.43) POLBCA12CA1CA2CA9
SCHEMBL4488885 0.78 ALDH1A1 (0.52) DHFRMAPTGAA
SCHEMBL5149849 0.69 MAPT (0.57) POLBCA12CA1CA2CA9
SCHEMBL12495756 0.68 KDM4E (0.54) POLBCA12CA1CA2CA9
Bromide SCHEMBL21382416 0.68 MAPT (0.60) POLBCA12CA1CA2CA9
SCHEMBL10569845 0.67 LMNA (0.53) DHFRPOLBCA12CA1CA2
SCHEMBL4834106 0.66 ALDH1A1 (0.50) POLBMAPTGAAIDO1LOXL2
SCHEMBL28907414 0.66 POLB (0.53) POLBCA12CA1CA2CA9
SCHEMBL30041078 0.66 POLB (0.53) POLBCA12CA1CA2CA9
SCHEMBL28756594 0.65 CA1 (0.60) CA1CA2CA9MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7560552-B2 Thiopyrimidine and isothiazolopyrimidine kinase inhibitors ABBOTT LABORATORIES (US) 2009-07-14 US disclosed