SCHEMBL13788838

SCHEMBL13788838

COc1cc(C(C)C)cc(O)c1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.44
GABRB2 P47870 1/20 0.44
TRPA1 O75762 1/20 0.44
PTGS1 P23219 1/20 0.44
CACNA1C Q13936 1/20 0.44
CYP3A4 P08684 3/20 0.43
TUBB4A P04350 2/20 0.41
TUBB P07437 2/20 0.41
TUBA3C P0DPH7 2/20 0.41
TUBA1B P68363 2/20 0.41
TUBA4A P68366 2/20 0.41
TUBB4B P68371 2/20 0.41
TUBB3 Q13509 2/20 0.41
TUBB2A Q13885 2/20 0.41
TUBB8 Q3ZCM7 2/20 0.41
TUBA3E Q6PEY2 2/20 0.41
TUBA1A Q71U36 2/20 0.41
TUBA1C Q9BQE3 2/20 0.41
TUBB6 Q9BUF5 2/20 0.41
TUBB2B Q9BVA1 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11436435 0.85 HDAC4 (0.44) CYP3A4HDAC4HDAC8
SCHEMBL20131281 0.83 GABRA1 (0.57) GABRA1GABRB2TRPA1PTGS1CACNA1C
SCHEMBL1494320 0.80 TRPA1 (0.56) GABRA1GABRB2TRPA1PTGS1CACNA1C
SCHEMBL13788860 0.80 TUBB1 (0.53) GABRA1GABRB2TRPA1PTGS1CACNA1C
SCHEMBL31545189 0.80 GABRA1 (0.44) GABRA1GABRB2TRPA1PTGS1CACNA1C
SCHEMBL17084596 0.79 HDAC4 (0.40) CYP3A4TUBB1HDAC4HDAC8
SCHEMBL6243516 0.79 PKM (0.48) GABRA1GABRB2PTGS1CYP3A4HDAC4
SCHEMBL12137640 0.76 EGFR (0.44) GABRA1GABRB2TRPA1PTGS1CACNA1C
SCHEMBL12360643 0.76 HDAC4 (0.38) GABRA1GABRB2CYP3A4TUBB1HDAC4
SCHEMBL19726452 0.76 HDAC4 (0.38) CYP3A4TSHRNFKB1HDAC4HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7557207-B2 Spiro 2,4-pyrimidinediamine compounds and their uses RIGEL PHARMACEUTICALS, INC. (US) 2009-07-07 US disclosed