SCHEMBL13797604

SCHEMBL13797604

CC(C)c1ccc(NC(=O)C(F)(F)C(F)(F)C(F)(F)F)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 8/20 0.51
HDAC7 Q8WUI4 8/20 0.51
HDAC8 Q9BY41 8/20 0.51
HDAC6 Q9UBN7 7/20 0.51
CA1 P00915 3/20 0.51
CA2 P00918 3/20 0.51
ALDH1A1 P00352 2/20 0.49
KIF11 P52732 1/20 0.49
PDK1 Q15118 1/20 0.46
PDK2 Q15119 1/20 0.46
PDK3 Q15120 1/20 0.46
PDK4 Q16654 1/20 0.46
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46
HDAC9 Q9UKV0 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46
HPGD P15428 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11097805 0.83 KIF11 (0.54) CA1CA2ALDH1A1KIF11PDK1
SCHEMBL29091743 0.81 KIF11 (0.53) CA1CA2ALDH1A1KIF11PDK1
SCHEMBL26624042 0.80 CA1 (0.56) HDAC1HDAC7HDAC8HDAC6CA1
SCHEMBL17577313 0.80 CA1 (0.56) HDAC1HDAC7HDAC8HDAC6CA1
SCHEMBL10646962 0.79 CA1 (0.41) HDAC1HDAC7HDAC8HDAC6CA1
SCHEMBL8846991 0.78 HDAC1 (0.72) HDAC1HDAC7HDAC8HDAC6CA1
SCHEMBL12788587 0.78 L3MBTL1 (0.73) CA1CA2ALDH1A1KIF11HPGD
SCHEMBL11036752 0.76 HPGD (0.56) CA1CA2ALDH1A1KIF11HPGD
SCHEMBL26623072 0.75 MDM2 (0.52) HDAC1HDAC7HDAC8HDAC6CA1
SCHEMBL10648232 0.74 HDAC1 (0.76) HDAC1HDAC7HDAC8HDAC6CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7550458-B2 Tricycloundecane compounds useful as modulators of nuclear hormone receptor function BRISTOL-MYERS SQUIBB COMPANY (US) 2009-06-23 US disclosed
US-7550458-B2 Tricycloundecane compounds useful as modulators of nuclear hormone receptor function BRISTOL-MYERS SQUIBB COMPANY (US) 2009-06-23 US disclosed