SCHEMBL1380290

SCHEMBL1380290

Cc1cc(F)cc2c(=O)[nH]c(=O)n(C3CC3)c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EEF2K O00418 1/20 0.39
TNKS O95271 6/20 0.38
PARP1 P09874 4/20 0.38
TNKS2 Q9H2K2 4/20 0.38
KCNH2 Q12809 3/20 0.37
CHRM1 P11229 3/20 0.36
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM5 P08912 1/20 0.36
CHRM3 P20309 1/20 0.36
JAK2 O60674 3/20 0.36
JAK1 P23458 3/20 0.36
JAK3 P52333 3/20 0.36
TYK2 P29597 2/20 0.36
ALDH1A1 P00352 3/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7559739 0.99 TNKS (0.38) EEF2KTNKSPARP1TNKS2KCNH2
SCHEMBL6644175 0.82 ALDH1A1 (0.44) EEF2KTNKSJAK2JAK1JAK3
Hydrochloric Acid SCHEMBL7556675 0.81 ALDH1A1 (0.43) EEF2KTNKSJAK2JAK1JAK3
SCHEMBL4505813 0.79 TOP2A (0.39) EEF2KKCNH2CHRM1CHRM2CHRM4
SCHEMBL6646396 0.77 EEF2K (0.37) EEF2KKCNH2CHRM1CHRM2CHRM4
SCHEMBL6668566 0.77 EEF2K (0.37) EEF2KKCNH2CHRM1CHRM2CHRM4
SCHEMBL1383138 0.77 PARP1 (0.40) EEF2KPARP1CHRM1CHRM2CHRM4
SCHEMBL6670008 0.75 JAK2 (0.39) EEF2KKCNH2CHRM1CHRM2CHRM4
SCHEMBL1381428 0.74 OPRM1 (0.45) EEF2KTNKSPARP1CHRM1HSD11B1
SCHEMBL12835810 0.73 EEF2K (0.41) EEF2KJAK2JAK1JAK3TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4811978-B2 2011-11-09 JP claimed
EP-1401830-A2 QUINAZOLINEDIONES AS ANTIBACTERIAL AGENTS Warner-Lambert Company LLC (US) 2004-03-31 EP claimed
WO-2002102793-A2 QUINAZOLINEDIONES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY LLC (US) 2002-12-27 WO claimed
EP-1255739-A1 3-AMINOQUINAZOLIN-2,4-DIONE ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 2002-11-13 EP claimed
WO-2001053273-A1 3-AMINOQUINAZOLIN-2,4-DIONE ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 2001-07-26 WO claimed