SCHEMBL13809017

SCHEMBL13809017

Cc1ccc(C(=O)N2CCc3cc4c(cc3C2c2ccccn2)OCO4)c(C(=O)O)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.50
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
HHAT Q5VTY9 1/20 0.40
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 3/20 0.38
HPGD P15428 3/20 0.38
GLA P06280 2/20 0.38
CASP1 P29466 2/20 0.38
CASP7 P55210 2/20 0.38
HSD17B10 Q99714 2/20 0.38
CYP2D6 P10635 1/20 0.38
GRIN2C Q14957 1/20 0.37
GAA P10253 2/20 0.37
TDP1 Q9NUW8 1/20 0.36
TRPC3 Q13507 1/20 0.35
TRPC6 Q9Y210 1/20 0.35
MAPT P10636 3/20 0.35
TSHR P16473 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13748721 0.95 MEN1 (0.44) KIF11MEN1KMT2AHHATKDM4E
SCHEMBL13809014 0.91 KIF11 (0.48) KIF11HHATKDM4EALDH1A1HPGD
SCHEMBL13809015 0.88 KIF11 (0.45) KIF11HHATKDM4EALDH1A1HPGD
SCHEMBL13809243 0.81 KIF11 (0.53) KIF11MEN1KMT2AKDM4EALDH1A1
SCHEMBL13809005 0.70 KIF11 (0.50) KIF11KMT2AKDM4EALDH1A1HPGD
SCHEMBL11718509 0.66 KIF11 (0.59) KIF11KDM4EALDH1A1HPGDGLA
SCHEMBL13822114 0.62 HCRTR1 (0.33) KIF11MEN1KMT2AMAPT
SCHEMBL10025892 0.62 P2RX7 (0.39) GRIN2C
SCHEMBL13748143 0.62 MAPT (0.75) KDM4EALDH1A1GAATDP1MAPT
SCHEMBL13748440 0.61 MAPT (0.66) KDM4EALDH1A1GAATDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009073545-A2 TETRAHYDRO-ISOQUINOLINE PPAT INHIBITORS AS ANTIBACTERIAL AGENTS MAXTHERA, INC. (US) 2009-06-11 WO disclosed