SCHEMBL13809227

SCHEMBL13809227

COc1cc2c(c(OC)c1)C(c1cccc(F)c1F)N(C(=O)c1ccc(-c3nnn[nH]3)cc1)CC2

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRIN2C Q14957 4/20 0.43
KMT2A Q03164 4/20 0.42
MEN1 O00255 3/20 0.42
CA12 O43570 3/20 0.40
CA1 P00915 3/20 0.40
CA2 P00918 3/20 0.40
CA7 P43166 3/20 0.40
CA9 Q16790 3/20 0.40
CA14 Q9ULX7 3/20 0.40
LMNA P02545 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
ABCB1 P08183 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.39
TP53 P04637 2/20 0.38
MTNR1B P49286 1/20 0.37
ROCK2 O75116 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13809233 0.93 GRIN2C (0.43) GRIN2CKMT2AMEN1LMNAMTNR1B
SCHEMBL13809246 0.82 GRIN2C (0.51) GRIN2CKMT2AMEN1CA12CA1
SCHEMBL13809247 0.80 GRIN2C (0.49) GRIN2CKMT2AMEN1CA12CA1
SCHEMBL13809019 0.75 GRIN2C (0.44) GRIN2CKMT2AMEN1LMNATP53
SCHEMBL13809245 0.75 RXFP1 (0.45) GRIN2CKMT2AMEN1LMNATP53
SCHEMBL4552564 0.71 GRIN2C (0.64) GRIN2CKMT2AMEN1CA12CA1
SCHEMBL4423052 0.70 GRIN2C (0.57) GRIN2CKMT2AMEN1CA12CA1
SCHEMBL4413383 0.69 KMT2A (0.47) GRIN2CKMT2AMEN1CA12CA1
SCHEMBL4414785 0.69 GRIN2C (0.54) GRIN2CKMT2AMEN1CA12CA1
SCHEMBL4415216 0.69 GRIN2C (0.55) GRIN2CKMT2AMEN1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009073545-A2 TETRAHYDRO-ISOQUINOLINE PPAT INHIBITORS AS ANTIBACTERIAL AGENTS MAXTHERA, INC. (US) 2009-06-11 WO disclosed