SCHEMBL13809245

SCHEMBL13809245

COc1cc2c(c(OC)c1)C(c1cccc(F)c1F)N(C(=O)c1ccccc1C#N)CC2

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 2/20 0.45
TP53 P04637 1/20 0.45
GRIN2C Q14957 5/20 0.45
LMNA P02545 1/20 0.42
MTNR1B P49286 1/20 0.42
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13809246 0.86 GRIN2C (0.51) TP53GRIN2CLMNAMEN1KMT2A
SCHEMBL13809019 0.82 GRIN2C (0.44) RXFP1TP53GRIN2CLMNAMTNR1B
SCHEMBL13809247 0.78 GRIN2C (0.49) TP53GRIN2CLMNAMEN1KMT2A
SCHEMBL13809227 0.75 GRIN2C (0.43) TP53GRIN2CLMNAMTNR1BMEN1
SCHEMBL13809233 0.74 GRIN2C (0.43) GRIN2CLMNAMTNR1BMEN1KMT2A
SCHEMBL13809251 0.71 GRIN2C (0.49) GRIN2CLMNAMTNR1BMEN1KMT2A
SCHEMBL13809228 0.71 GRIN2C (0.43) GRIN2CMEN1KMT2A
SCHEMBL4422963 0.70 GRIN2C (0.47) GRIN2CLMNAMTNR1BMEN1KMT2A
SCHEMBL4424076 0.69 GRIN2C (0.45) RXFP1TP53GRIN2CMTNR1BMEN1
SCHEMBL4421922 0.68 KMT2A (0.46) RXFP1TP53GRIN2CMTNR1BMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009073545-A2 TETRAHYDRO-ISOQUINOLINE PPAT INHIBITORS AS ANTIBACTERIAL AGENTS MAXTHERA, INC. (US) 2009-06-11 WO disclosed