SCHEMBL13809247

SCHEMBL13809247

COc1cc2c(c(OC)c1)C(c1cccc(F)c1F)N(C(=O)c1ccc(Cl)nc1)CC2

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRIN2C Q14957 9/20 0.49
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
LMNA P02545 2/20 0.42
CA12 O43570 3/20 0.41
CA1 P00915 3/20 0.41
CA2 P00918 3/20 0.41
CA7 P43166 3/20 0.41
CA9 Q16790 3/20 0.41
CA14 Q9ULX7 3/20 0.41
GRIN2D O15399 1/20 0.41
TP53 P04637 1/20 0.41
HPGD P15428 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13809246 0.83 GRIN2C (0.51) GRIN2CKMT2AMEN1LMNACA12
SCHEMBL13809019 0.82 GRIN2C (0.44) GRIN2CKMT2AMEN1LMNATP53
SCHEMBL13809227 0.80 GRIN2C (0.43) GRIN2CKMT2AMEN1LMNACA12
SCHEMBL13809233 0.78 GRIN2C (0.43) GRIN2CKMT2AMEN1LMNA
SCHEMBL13809245 0.78 RXFP1 (0.45) GRIN2CKMT2AMEN1LMNATP53
SCHEMBL4411776 0.72 NPC1 (0.53) GRIN2CKMT2AMEN1CA12CA1
SCHEMBL13809240 0.72 GRIN2C (0.54) GRIN2CKMT2AMEN1GRIN2D
SCHEMBL13809251 0.71 GRIN2C (0.49) GRIN2CKMT2AMEN1LMNACA12
SCHEMBL4413383 0.70 KMT2A (0.47) GRIN2CKMT2AMEN1LMNACA12
SCHEMBL4422268 0.70 GRIN2C (0.55) GRIN2CKMT2AMEN1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009073545-A2 TETRAHYDRO-ISOQUINOLINE PPAT INHIBITORS AS ANTIBACTERIAL AGENTS MAXTHERA, INC. (US) 2009-06-11 WO disclosed