SCHEMBL13811458

SCHEMBL13811458

COC(=O)C1=NOC2(CCN(C(=O)OC(C)(C)C)CC2)C1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 2/20 0.57
PKM P14618 1/20 0.42
ALOX15 P16050 2/20 0.42
TP53 P04637 1/20 0.42
MAPT P10636 1/20 0.42
HSD17B10 Q99714 1/20 0.42
USP2 O75604 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NR1H2 P55055 1/20 0.40
JAK2 O60674 1/20 0.38
JAK1 P23458 1/20 0.38
SCD5 Q86SK9 1/20 0.38
TSHR P16473 1/20 0.37
ATM Q13315 1/20 0.37
EPHX2 P34913 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1639199 0.88 GPR119 (0.57) GPR119ALOX15TP53MAPTHSD17B10
SCHEMBL2401311 0.86 GPR119 (0.52) GPR119ALOX15TP53MAPTHSD17B10
SCHEMBL31470380 0.84 GPR119 (0.53) GPR119ALOX15TP53MAPTHSD17B10
SCHEMBL31470348 0.83 GPR119 (0.48) GPR119ALOX15TP53MAPTHSD17B10
SCHEMBL13170189 0.81 GPR119 (0.50) GPR119USP2SMN1; SMN2SCD5
SCHEMBL23097412 0.81 MAPT (0.40) GPR119MAPTHSD17B10
SCHEMBL12901469 0.80 GPR119 (0.49) GPR119PKMUSP2SMN1; SMN2
SCHEMBL12901537 0.80 GPR119 (0.49) GPR119USP2SMN1; SMN2
SCHEMBL31470342 0.80 GPR119 (0.50) GPR119PKMALOX15TP53MAPT
SCHEMBL2599806 0.79 PKM (0.55) GPR119PKMJAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954698-B1 SPIROCYCLIC COMPOUNDS AS HDAC INHIBITORS MERCK & CO INC (US) 2009-06-24 EP disclosed