SCHEMBL1381906

SCHEMBL1381906

C=C(C(N)=O)c1ccc(Cl)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.52
CES1 P23141 3/20 0.52
ALOX15 P16050 1/20 0.50
TSHR P16473 1/20 0.50
LMNA P02545 3/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
MAPT P10636 1/20 0.48
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
NPC1 O15118 2/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
GSK3B P49841 2/20 0.45
SRD5A2 P31213 1/20 0.45
MAPK1 P28482 1/20 0.45
MAOA P21397 2/20 0.44
MAOB P27338 2/20 0.44
CYP1A2 P05177 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5781080 0.94 MAP4K4 (0.50) CES2CES1ALOX15TSHRLMNA
SCHEMBL9864000 0.89 PARP10 (0.52) ALDH1A1MAPTRAB9AMAOAMAOB
SCHEMBL1450228 0.88 PARP10 (0.39) TSHRLMNAL3MBTL1ALDH1A1MAPT
SCHEMBL11699267 0.82 ALDH1A1 (0.42) CES2CES1ALOX15TSHRLMNA
SCHEMBL2081411 0.80 CES2 (0.52) CES2CES1ALOX15TSHRLMNA
SCHEMBL126170 0.79 ALOX15 (0.58) CES2CES1ALOX15TSHRLMNA
SCHEMBL11798461 0.79 PARP10 (0.47) ALOX15TSHRLMNAKDM4EALDH1A1
SCHEMBL6203654 0.79 CES2 (0.68) CES2CES1ALOX15TSHRLMNA
SCHEMBL10552849 0.79 CES2 (0.54) CES2CES1ALOX15TSHRLMNA
SCHEMBL1033882 0.79 TSHR (0.57) CES2CES1ALOX15TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3921317-A1 3-AMINO-2-[2-(ACYLAMINO)PYRIDIN-4-YL]-1,5,6,7-TETRAHYDRO-4H-PYRROLO[3,2-C]PYRIDIN-4-ONE AS CSNK1 INHIBITORS Bayer Aktiengesellschaft (DE) 2021-12-15 EP claimed
WO-2020161257-A1 3-AMINO-2-[2-(ACYLAMINO)PYRIDIN-4-YL]-1,5,6,7-TETRAHYDRO-4H-PYRROLO[3,2-C]PYRIDIN-4-ONE AS CSNK1 INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2020-08-13 WO claimed
CN-110124735-A A kind of hydrophilic electroconductive hydrogel cathode catalysis film and its preparation method and application 中钢集团鞍山热能研究院有限公司 2019-08-16 CN claimed
JP-4828407-B2 2011-11-30 JP claimed
EP-1594869-A2 3-SUBSTITUTED-2(ARYLALKYL)-1-AZABICYCLOALKANES AND METHODS OF USE THEREOF Targacept, Inc. (US) 2005-11-16 EP claimed
WO-2004076449-A2 3-SUBSTITUTED-2(ARYLALKYL)-1-AZABICYCLOALKANES AND METHODS OF USE THEREOF TARGACEPT, INC. (US) 2004-09-10 WO claimed
CN-118955381-A Pyrazole compound as well as preparation method and application thereof 赣南师范大学 2024-11-15 CN disclosed
CN-117219278-A Schizophrenia aggressive behavior risk assessment model and application thereof 福建省立医院 2023-12-12 CN disclosed
CN-117191993-A Metabolic biomarker for aggressive behavior of schizophrenia and screening method thereof 郑富豪 2023-12-08 CN disclosed
CN-110124735-A A kind of hydrophilic electroconductive hydrogel cathode catalysis film and its preparation method and application 中钢集团鞍山热能研究院有限公司 2019-08-16 CN disclosed
US-20160272600-A1 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, LLC 2016-09-22 US disclosed
US-20070042275-A1 Composition for optical recording, optical recording medium, and production method thereof FUJI PHOTO FILM CO., LTD. 2007-02-22 US disclosed
US-4302484-A Polymers crosslinkable by electron beams BAYER AKTIENGESELLSCHAFT (DE) 1981-11-24 US disclosed
EP-0001997-B1 ELECTRON BEAM-CURABLE PHOTORESIST LACQUERS BAYER AG (DE) 1981-02-11 EP disclosed
EP-0001997-A1 Electron beam-curable photoresist lacquers BAYER AG (DE) 1979-05-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160272600-A1 INHIBITORS OF BETA-SECRETASE BACE1, BACE2, PSEN1 CES2 943/4885CES1 361/4885ALOX15 2821/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.