SCHEMBL13822828

SCHEMBL13822828

CC(C)c1ccc(N)c(NC(=O)c2cc3c(s2)CN(C(=O)O)CC3)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 4/20 0.47
ALDH1A1 P00352 5/20 0.40
HPGD P15428 4/20 0.40
TP53 P04637 2/20 0.40
MAPK1 P28482 1/20 0.40
KDM1A O60341 1/20 0.39
RAB9A P51151 6/20 0.39
KDM4E B2RXH2 3/20 0.39
NPSR1 Q6W5P4 2/20 0.39
HDAC2 Q92769 2/20 0.38
MAPT P10636 5/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
PLA2G1B P04054 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
ATG4B Q9Y4P1 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
NPC1 O15118 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL979002 0.85 NPC1 (0.48) HDAC6ALDH1A1KDM1ARAB9AHDAC2
SCHEMBL13822878 0.84 KDM1A (0.51) HDAC6ALDH1A1HPGDMAPK1KDM1A
SCHEMBL975199 0.83 L3MBTL1 (0.44) HDAC6ALDH1A1HPGDRAB9AKDM4E
SCHEMBL978070 0.83 HTR2C (0.52) RAB9AHDAC2MAPTKMT2AMEN1
SCHEMBL975053 0.82 SMN1; SMN2 (0.41) HDAC6ALDH1A1HPGDRAB9AKDM4E
SCHEMBL976172 0.81 MEN1 (0.45) HDAC6ALDH1A1HPGDKDM1ARAB9A
SCHEMBL978288 0.81 ALDH1A1 (0.43) HDAC6ALDH1A1KDM1ARAB9AKDM4E
SCHEMBL13822812 0.76 KDM1A (0.60) HDAC6ALDH1A1HPGDMAPK1KDM1A
SCHEMBL1175185 0.74 RAB9A (0.60) HDAC6ALDH1A1TP53MAPK1RAB9A
SCHEMBL13822935 0.74 MAPT (0.37) HDAC6ALDH1A1TP53KDM4EHDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2197552-B1 NOVEL TETRAHYDROFUSEDPYRIDINES AS HISTONE DEACETYLASE INHIBITORS 4SC AG (DE) 2012-11-21 EP claimed