SCHEMBL13824906

SCHEMBL13824906

O=c1[nH]nc2c(COCc3ccccc3)cc(-c3ccccc3)cn12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RET P07949 1/20 0.42
MET P08581 1/20 0.42
LTK P29376 1/20 0.42
GRK5 P34947 1/20 0.42
CDK8 P49336 1/20 0.42
RPS6KA3 P51812 1/20 0.42
MST1R Q04912 1/20 0.42
TYRO3 Q06418 1/20 0.42
DYRK1A Q13627 1/20 0.42
LRRK2 Q5S007 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
ALK Q9UM73 1/20 0.42
DYRK1B Q9Y463 1/20 0.42
PDE5A O76074 2/20 0.41
PDE3B Q13370 2/20 0.38
PDE3A Q14432 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13824909 0.81 LTK (0.50) RETMETLTKGRK5CDK8
SCHEMBL13825028 0.71 LTK (0.48) RETMETLTKGRK5CDK8
SCHEMBL13825030 0.69 LTK (0.46) RETMETLTKGRK5CDK8
SCHEMBL13825035 0.69 HPGDS (0.48) PDE3BPDE3AL3MBTL1NPC1RAB9A
SCHEMBL2513747 0.66 TSHR (0.47) L3MBTL1NPC1RAB9ATSHRALDH1A1
Biphenyl SCHEMBL1702724 0.66 TSHR (0.83) TSHRHSP90AB1ALDH1A1KDM4E
SCHEMBL22593160 0.65 TSHR (0.46) L3MBTL1NPC1RAB9ATSHRADORA3
SCHEMBL18632535 0.64 SCN5A (0.62) RETMETLTKGRK5CDK8
SCHEMBL18632530 0.64 SCN5A (0.62) RETMETLTKGRK5CDK8
SCHEMBL22322658 0.63 KMT2A (0.44) L3MBTL1NPC1RAB9ATSHRADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012150829-A2 NOBLE TRIAZOLOPYRIDINE DERIVATIVE OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF, PRODUCTION METHOD THEREOF, AND PHARMACEUTICAL COMPOSITION INCLUDING SAME 제일약품주식회사 (KR) 2012-11-08 WO disclosed