SCHEMBL13824910

SCHEMBL13824910

CNc1c(NCC2CC2)ccc(OS(=O)(=O)C(F)(F)F)c1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LIPC P11150 1/20 0.40
LIPG Q9Y5X9 1/20 0.40
CNR2 P34972 4/20 0.36
CNR1 P21554 3/20 0.36
DRD2 P14416 5/20 0.34
DRD3 P35462 5/20 0.34
DRD4 P21917 3/20 0.34
HTR1D P28221 2/20 0.34
DRD1 P21728 2/20 0.34
DRD5 P21918 2/20 0.34
HTR5A P47898 1/20 0.34
BRD4 O60885 2/20 0.33
PTGER4 P35408 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18374895 0.69 DRD2 (0.35) DRD2DRD3DRD4HTR1DDRD1
SCHEMBL17340574 0.67 DRD2 (0.35) DRD2DRD3DRD4HTR1DDRD1
SCHEMBL13726636 0.65 GRM2 (0.51) DRD2DRD3DRD4DRD1DRD5
SCHEMBL18364503 0.63 DRD2 (0.33) DRD2DRD3DRD4HTR1DDRD1
SCHEMBL25027141 0.62 DRD2 (0.38) LIPCLIPGDRD2DRD3DRD4
SCHEMBL15586261 0.61 DRD2 (0.43) DRD2DRD3DRD4HTR1DDRD1
SCHEMBL19948194 0.61 DRD2 (0.41) DRD2DRD3DRD4HTR1DDRD1
SCHEMBL3997164 0.60 ALDH1A1 (0.65) BRD4PTGER4
SCHEMBL16006621 0.60 DRD2 (0.44) DRD2DRD3DRD4HTR1DDRD1
SCHEMBL3997818 0.59 ALDH1A1 (0.53) LIPCLIPGCNR2CNR1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012151139-A1 ALKYNE BENZOTRIAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-11-08 WO disclosed