SCHEMBL13827487

SCHEMBL13827487

CCCS(=O)(=O)NCCOc1cc2c(cc1F)CCCNC2Cc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 6/20 0.41
CYP3A4 P08684 1/20 0.41
KDM1A O60341 1/20 0.40
ADRB2 P07550 1/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13827488 0.94 KDM1A (0.42) SLC6A9KDM1AADRB2KDM4EGAA
SCHEMBL13736151 0.89 SLC6A9 (0.48) SLC6A9KDM1AADRB2KDM4EGAA
SCHEMBL13827430 0.85 SLC6A9 (0.56) SLC6A9CYP3A4KCNH2
SCHEMBL13827500 0.83 SLC6A9 (0.44) SLC6A9KDM1AADRB2
SCHEMBL15187753 0.83 SLC6A9 (0.40) SLC6A9KDM1AADRB2KDM4EGAA
SCHEMBL17675759 0.82 SLC6A9 (0.53) SLC6A9GAABCHEACHEKCNH2
SCHEMBL13737473 0.81 ADRB2 (0.48) KDM1AADRB2KDM4EGAAMAPT
SCHEMBL17675711 0.80 SLC6A9 (0.55) SLC6A9CYP3A4BCHEACHEKCNH2
SCHEMBL17675761 0.80 SLC6A9 (0.53) SLC6A9CYP3A4KCNH2
SCHEMBL13827332 0.79 SLC6A9 (0.56) SLC6A9CYP3A4ADRB2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9309200-B2 Benzazepine derivatives, pharmaceutical compositions containing them, and their use in therapy AbbVie Deutschland GmbH & Co. KG (DE) 2016-04-12 US disclosed
US-9309200-B2 Benzazepine derivatives, pharmaceutical compositions containing them, and their use in therapy AbbVie Deutschland GmbH & Co. KG (DE) 2016-04-12 US disclosed
WO-2012152915-A1 BENZAZEPINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, AND THEIR USE IN THERAPY ABBOTT GMBH & CO. KG (DE) 2012-11-15 WO disclosed