SCHEMBL1383289

SCHEMBL1383289

NC(=O)c1cccc(Cc2cc3ccccc3[nH]2)c1N1CCCCC1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.44
HRH3 Q9Y5N1 1/20 0.43
PARP1 P09874 7/20 0.43
AHR P35869 2/20 0.41
PLAU P00749 1/20 0.40
KDM4E B2RXH2 1/20 0.39
HSD17B10 Q99714 1/20 0.39
LOXL2 Q9Y4K0 1/20 0.39
CCKAR P32238 1/20 0.39
PCSK9 Q8NBP7 3/20 0.38
KDR P35968 1/20 0.38
F2 P00734 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7077495 0.82 AHR (0.51) PARP1AHRKDM4EHSD17B10LOXL2
SCHEMBL23632367 0.77 NPC1 (0.50) NPC1PARP1KDM4EHSD17B10
SCHEMBL28046983 0.75 NPC1 (0.54) NPC1PARP1KDM4EHSD17B10
SCHEMBL1382512 0.74 CHEK2 (0.45) PARP1AHRKDM4ELOXL2PCSK9
SCHEMBL3681824 0.73 NPC1 (0.66) NPC1PARP1KDM4EHSD17B10
SCHEMBL29990403 0.73 MTNR1A (0.51) HRH3PARP1AHRKDM4EHSD17B10
SCHEMBL3682185 0.72 NPC1 (0.62) NPC1PARP1KDM4EHSD17B10
Urea SCHEMBL28780664 0.70 PLAU (0.48) NPC1HRH3PLAUKDM4EHSD17B10
SCHEMBL1383288 0.70 NPC1 (0.48) NPC1HRH3KDM4EHSD17B10CCKAR
SCHEMBL19667085 0.70 NPC1 (0.47) NPC1PARP1KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4831907-B2 2011-12-07 JP claimed
EP-1225894-A4 FAB I INHIBITORS SMITHKLINE BEECHAM CORP (US) 2003-01-08 EP claimed
EP-1225894-A1 FAB I INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2002-07-31 EP claimed
WO-2001026652-A1 FAB I INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-04-19 WO claimed
EP-1225894-A4 FAB I INHIBITORS SMITHKLINE BEECHAM CORP (US) 2003-01-08 EP disclosed
EP-1225894-A1 FAB I INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2002-07-31 EP disclosed
WO-2001026652-A1 FAB I INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-04-19 WO disclosed