SCHEMBL13837397

SCHEMBL13837397

CC(C)(C)OC(=O)N1CCC(COc2ccc(-c3ccc(F)cc3)cc2)C1

nearest known ligand 0.82

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 11/20 0.52
CHEK2 O96017 2/20 0.51
HDAC1 Q13547 1/20 0.50
HDAC2 Q92769 1/20 0.50
ALOX5AP P20292 2/20 0.49
FEN1 P39748 2/20 0.49
MMP13 P45452 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1769253 0.90 CHEK2 (0.56) GPR119CHEK2ALOX5APFEN1
SCHEMBL1769099 0.90 GPR119 (0.57) GPR119CHEK2
SCHEMBL19610292 0.86 GPR119 (0.54) GPR119CHEK2ALOX5APFEN1
SCHEMBL22756382 0.85 GPR119 (0.56) GPR119CHEK2ALOX5APFEN1
SCHEMBL26311640 0.85 GPR119 (0.53) GPR119CHEK2HDAC1ALOX5APFEN1
SCHEMBL21398088 0.85 GPR119 (0.53) GPR119CHEK2HDAC1ALOX5APFEN1
SCHEMBL14006542 0.85 GPR119 (0.53) GPR119CHEK2ALOX5APFEN1
SCHEMBL31071572 0.85 GPR119 (0.53) GPR119CHEK2
SCHEMBL13876978 0.85 KDM4E (0.56) GPR119
SCHEMBL31330775 0.84 GPR119 (0.54) GPR119CHEK2HDAC1ALOX5APFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9000010-B2 Alkyl-heterocycle carbamate derivatives, their preparation and their therapeutic application SANOFI (FR) 2015-04-07 US disclosed
EP-2526100-B1 ALKYL-HETEROCYCLE CARBAMATE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION SANOFI SA (FR) 2013-12-04 EP disclosed
US-20120295909-A1 ALKYL-HETEROCYCLE CARBAMATE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION SANOFI (FR) 2012-11-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120295909-A1 ALKYL-HETEROCYCLE CARBAMATE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION PRMT9, PRMT8, CBR1 GPR119 242/4885CHEK2 3802/4885HDAC1 125/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.