SCHEMBL13845405

SCHEMBL13845405

CC12C[C@H]3CC(OC(=O)N4Cc5ccccc5NC4=O)C[C@@H](C1)N32

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.71
BRD4 O60885 1/20 0.40
CREBBP Q92793 1/20 0.40
CHRM1 P11229 4/20 0.37
CHRM4 P08173 3/20 0.37
KCNH2 Q12809 1/20 0.34
CHRM2 P08172 3/20 0.34
CHRM5 P08912 3/20 0.34
CHRM3 P20309 3/20 0.34
HTR2C P28335 2/20 0.34
LMNA P02545 2/20 0.34
BLM P54132 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
ADRA2C P18825 1/20 0.34
ADRA1A P35348 1/20 0.34
HRH1 P35367 1/20 0.34
KMT2A Q03164 1/20 0.34
NFKB1 P19838 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL508185 0.84 ALOX15 (0.98) ALOX15CHRM1CHRM4CHRM2CHRM5
SCHEMBL29468680 0.84 ALOX15 (0.98) ALOX15CHRM1CHRM4CHRM2CHRM5
SCHEMBL29462345 0.84 ALOX15 (0.98) ALOX15CHRM1CHRM4CHRM2CHRM5
SCHEMBL508184 0.84 ALOX15 (0.98) ALOX15CHRM1CHRM4CHRM2CHRM5
SCHEMBL2824864 0.68 BRD4 (0.56) ALOX15BRD4CREBBPMEN1KMT2A
SCHEMBL9202802 0.64 ALOX15 (0.53) ALOX15BRD4CREBBP
SCHEMBL9198302 0.61 ALOX15 (0.50) ALOX15BRD4CREBBPCHRM1CHRM4
SCHEMBL2212650 0.60 CHRM4 (0.50) ALOX15CHRM1CHRM4
SCHEMBL22716676 0.60 MAPK1 (0.55) ALOX15BRD4CREBBPCHRM1CHRM4
SCHEMBL28355036 0.60 BRD4 (0.61) ALOX15BRD4CREBBPBLMKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009060203-A1 3,4,6,7-TETRAHYDRO-1 H-PYRROLO[3,4-D]PYRIMIDINE-2,5-DIONES AND THEIR THERAPEUTIC USE ARGENTA DISCOVERY LIMITED (GB) 2009-05-14 WO disclosed