SCHEMBL13848253

SCHEMBL13848253

Nc1ncc(-c2cc(NCCc3c[nH]c4ccccc34)nc(N3CCOCC3)n2)cn1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADK P55263 3/20 0.57
HTR1A P08908 1/20 0.54
DRD2 P14416 1/20 0.54
HTR2A P28223 1/20 0.54
HTR7 P34969 1/20 0.54
HTR6 P50406 1/20 0.54
PIK3CA P42336 13/20 0.54
PIK3CG P48736 3/20 0.51
PIK3R1 P27986 3/20 0.51
PIK3CB P42338 2/20 0.51
MTOR P42345 1/20 0.51
EIF2AK2 P19525 1/20 0.49
MAP3K12 Q12852 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4120692 0.84 PIK3CA (0.51) ADKHTR1ADRD2HTR2AHTR7
SCHEMBL13848003 0.83 PIK3CA (0.62) PIK3CAPIK3CGPIK3R1PIK3CBMTOR
SCHEMBL13848256 0.81 PIK3CA (0.73) PIK3CAPIK3CGPIK3R1PIK3CBMTOR
SCHEMBL13848242 0.79 PIK3CA (0.59) PIK3CAPIK3CGPIK3R1PIK3CBMTOR
SCHEMBL13848167 0.78 PIK3CA (0.69) PIK3CAPIK3CGPIK3R1PIK3CBMTOR
SCHEMBL13848181 0.78 PIK3CA (0.73) PIK3CAPIK3CGPIK3R1PIK3CBMTOR
SCHEMBL13848250 0.77 PIK3CA (0.65) PIK3CAPIK3CGPIK3R1PIK3CBMTOR
SCHEMBL10327936 0.75 PIK3CA (0.65) PIK3CAPIK3CGPIK3R1PIK3CBMTOR
SCHEMBL13848239 0.75 PIK3CA (0.72) PIK3CAPIK3CGPIK3R1PIK3CBMTOR
SCHEMBL4117117 0.74 HTR1A (0.47) ADKHTR1ADRD2HTR2AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009066084-A1 2 -MORPHOLINOPYRIMIDINES AND THEIR USE AS PI3 KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2009-05-28 WO disclosed