SCHEMBL4120692

SCHEMBL4120692

Nc1ncc(-c2cc(OCCc3c[nH]c4ccccc34)nc(N3CCOCC3)n2)cn1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 14/20 0.51
MTOR P42345 4/20 0.51
MAP3K12 Q12852 1/20 0.49
ADK P55263 3/20 0.48
HTR1A P08908 3/20 0.46
AKT1 P31749 3/20 0.46
PIK3CB P42338 3/20 0.45
PIK3CD O00329 2/20 0.45
PIK3R1 P27986 2/20 0.45
PIK3CG P48736 2/20 0.45
PI4KB Q9UBF8 1/20 0.45
DRD2 P14416 1/20 0.45
HTR2A P28223 1/20 0.45
HTR7 P34969 1/20 0.45
HTR6 P50406 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4117117 0.90 HTR1A (0.47) PIK3CAMTORADKHTR1AAKT1
SCHEMBL13848253 0.84 ADK (0.57) PIK3CAMTORMAP3K12ADKHTR1A
SCHEMBL3990409 0.82 PIK3CA (0.58) PIK3CAMTORMAP3K12AKT1PIK3CB
SCHEMBL3997060 0.80 PIK3CA (0.59) PIK3CAMTORMAP3K12AKT1PIK3CB
SCHEMBL13848126 0.78 PIK3CA (0.56) PIK3CAMTORMAP3K12AKT1PIK3CB
SCHEMBL13848119 0.78 PIK3CA (0.53) PIK3CAMTORMAP3K12AKT1PIK3CB
SCHEMBL13848198 0.77 PIK3CA (0.60) PIK3CAMTORMAP3K12AKT1PIK3CB
SCHEMBL10327867 0.76 PIK3CA (0.61) PIK3CAMTORMAP3K12PIK3CBPIK3CD
SCHEMBL3990236 0.75 PIK3CA (0.51) PIK3CAMTORMAP3K12AKT1PIK3CB
SCHEMBL4125340 0.75 PIK3CA (0.60) PIK3CAMTORMAP3K12PIK3CBPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009066084-A1 2 -MORPHOLINOPYRIMIDINES AND THEIR USE AS PI3 KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2009-05-28 WO disclosed