SCHEMBL13848490

SCHEMBL13848490

CCOC(=O)c1csc(Cc2c[nH]c3ccccc23)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.54
MAPT P10636 9/20 0.51
NPC1 O15118 4/20 0.51
RAB9A P51151 4/20 0.51
SMN1; SMN2 Q16637 4/20 0.50
CYP1A2 P05177 3/20 0.50
CYP3A4 P08684 3/20 0.50
CYP2C19 P33261 3/20 0.50
CYP2D6 P10635 2/20 0.50
CYP2C9 P11712 2/20 0.50
MEN1 O00255 5/20 0.49
KMT2A Q03164 5/20 0.49
ALDH1A1 P00352 3/20 0.48
KDM4E B2RXH2 1/20 0.48
HSP90AA1 P07900 1/20 0.48
POLB P06746 1/20 0.47
GPR84 Q9NQS5 2/20 0.46
AHR P35869 2/20 0.46
NR1I2 O75469 1/20 0.46
MMP1 P03956 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21366239 0.88 MAPT (0.63) MAPTCYP1A2CYP3A4CYP2C19CYP2D6
SCHEMBL22462565 0.80 MEN1 (0.77) PKMMAPTNPC1RAB9ASMN1; SMN2
SCHEMBL5216804 0.79 MAPT (0.67) PKMMAPTNPC1RAB9ASMN1; SMN2
SCHEMBL10918829 0.78 HDAC1 (0.60) MAPTNPC1RAB9ASMN1; SMN2CYP1A2
SCHEMBL5125370 0.74 RAB9A (0.49) PKMMAPTNPC1RAB9ASMN1; SMN2
SCHEMBL4722943 0.74 MAPT (0.52) PKMMAPTNPC1RAB9ASMN1; SMN2
SCHEMBL1246735 0.73 RAB9A (0.64) PKMMAPTNPC1RAB9ASMN1; SMN2
SCHEMBL21366323 0.72 GPR84 (0.54) MAPTCYP3A4CYP2C19CYP2D6MEN1
SCHEMBL2838509 0.72 RAB9A (0.62) PKMMAPTNPC1RAB9ASMN1; SMN2
SCHEMBL2838513 0.72 RAB9A (0.62) PKMMAPTNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1365760-B1 PREPARATIONS AND USE OF AN AH RECEPTOR LIGAND, 2-(1'H-INDOLE-3'-CARBONYL)-THIAZOLE-4-CARBOXYLIC ACID METHYL ESTER WISCONSIN ALUMNI RES FOUND (US) 2009-05-20 EP disclosed