SCHEMBL13864591

SCHEMBL13864591

CC(=O)c1ccc(-c2ccc(O)cc2F)cc1

nearest known ligand 0.68

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 4/20 0.68
ESR1 P03372 8/20 0.54
ESR2 Q92731 4/20 0.54
APP P05067 3/20 0.50
CYP2C19 P33261 3/20 0.50
CYP2C9 P11712 2/20 0.50
CYP3A4 P08684 2/20 0.50
KIF11 P52732 1/20 0.47
CYP2D6 P10635 1/20 0.46
HSD17B2 P37059 1/20 0.45
PTGS1 P23219 1/20 0.45
MAPT P10636 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10436026 0.84 MAOB (0.55) HSD17B1APPCYP2C19CYP2C9CYP3A4
SCHEMBL30747689 0.84 MAOB (0.55) HSD17B1APPCYP2C19CYP2C9CYP3A4
SCHEMBL10925015 0.83 HSD17B1 (0.54) HSD17B1APPKIF11PTGS1MAPT
SCHEMBL2559215 0.83 RARB (0.59) HSD17B1APPCYP2C19CYP2C9CYP3A4
SCHEMBL497922 0.82 CA12 (0.58) HSD17B1ESR1ESR2APPCYP2C19
SCHEMBL5549813 0.81 MMP1 (0.49) HSD17B1APPKIF11PTGS1MAPT
SCHEMBL38659424 0.81 ESR1 (0.70) HSD17B1ESR1ESR2APPCYP2C19
SCHEMBL28226426 0.81 ESR1 (0.70) HSD17B1ESR1ESR2APPCYP2C19
SCHEMBL4101247 0.81 HSD17B1 (1.00) HSD17B1ESR1ESR2HSD17B2MAPT
SCHEMBL10922772 0.79 RARB (0.52) HSD17B1KIF11PTGS1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1479671-B1 Pyrimidinone compounds SMITHKLINE BEECHAM PLC (GB) 2009-05-27 EP disclosed