SCHEMBL13865720

SCHEMBL13865720

Cc1nccc2c(NC(=O)NC3CCN(c4ncccc4Cl)CC3)cccc12

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PAK1 Q13153 2/20 0.50
MALT1 Q9UDY8 9/20 0.48
TSHR P16473 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
TRPV1 Q8NER1 3/20 0.46
EPHX2 P34913 1/20 0.45
SIGMAR1 Q99720 1/20 0.43
KDM4E B2RXH2 1/20 0.43
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA4 P22748 2/20 0.43
CA7 P43166 2/20 0.43
CA9 Q16790 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13870115 0.90 PAK1 (0.49) PAK1MALT1TRPV1EPHX2SIGMAR1
SCHEMBL13865724 0.86 PAK1 (0.46) PAK1MALT1TSHRSMN1; SMN2TRPV1
SCHEMBL13865715 0.85 TRPV1 (0.54) PAK1TRPV1EPHX2SIGMAR1KDM4E
SCHEMBL13865684 0.84 CYP2C9 (0.49) PAK1SMN1; SMN2TRPV1KDM4E
SCHEMBL13865722 0.84 TRPV1 (0.45) PAK1TRPV1SIGMAR1KDM4ECA12
SCHEMBL13865712 0.84 PAK1 (0.46) PAK1SMN1; SMN2TRPV1KDM4E
SCHEMBL13865723 0.79 CCNC (0.43) PAK1TSHRSMN1; SMN2TRPV1SIGMAR1
SCHEMBL13865721 0.79 PAK1 (0.47) PAK1TRPV1EPHX2KDM4ECA12
SCHEMBL13865717 0.78 PAK1 (0.46) PAK1TRPV1SIGMAR1KDM4ECA12
SCHEMBL13865718 0.77 TRPV1 (0.47) PAK1TRPV1EPHX2KDM4ECA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7528151-B2 Heterocyclic urea derivatives for the treatment of pain GLAXO GROUP LIMITED (GB) 2009-05-05 US disclosed