SCHEMBL13865724

SCHEMBL13865724

COc1ccc(Cl)c(N2CCC(NC(=O)Nc3cccc4c(C)nccc34)CC2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAK1 Q13153 3/20 0.46
SIGMAR1 Q99720 1/20 0.42
KDM4E B2RXH2 1/20 0.42
CNR1 P21554 1/20 0.40
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MALT1 Q9UDY8 2/20 0.39
EPHX2 P34913 1/20 0.39
EPHX1 P07099 1/20 0.39
CA12 O43570 3/20 0.39
CA1 P00915 3/20 0.39
CA2 P00918 3/20 0.39
CA4 P22748 3/20 0.39
CA7 P43166 3/20 0.39
CA9 Q16790 3/20 0.39
CCNC P24863 1/20 0.39
CDK8 P49336 1/20 0.39
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39
TRPV1 Q8NER1 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13865725 0.88 TRPV1 (0.47) PAK1SIGMAR1KDM4EEPHX2TRPV1
SCHEMBL13865717 0.86 PAK1 (0.46) PAK1SIGMAR1KDM4EEPHX1CA12
SCHEMBL13865720 0.86 PAK1 (0.50) PAK1SIGMAR1KDM4ETSHRSMN1; SMN2
SCHEMBL13865722 0.85 TRPV1 (0.45) PAK1SIGMAR1KDM4ECNR1CA12
SCHEMBL13870115 0.80 PAK1 (0.49) PAK1SIGMAR1KDM4EMALT1EPHX2
SCHEMBL13865684 0.78 CYP2C9 (0.49) PAK1KDM4ESMN1; SMN2TRPV1
SCHEMBL13865723 0.78 CCNC (0.43) PAK1SIGMAR1KDM4ETSHRSMN1; SMN2
SCHEMBL13865712 0.78 PAK1 (0.46) PAK1KDM4ESMN1; SMN2TRPV1
SCHEMBL13865685 0.76 CLK2 (0.43) PAK1SIGMAR1KDM4EEPHX2EPHX1
SCHEMBL13865715 0.76 TRPV1 (0.54) PAK1SIGMAR1KDM4EEPHX2TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7528151-B2 Heterocyclic urea derivatives for the treatment of pain GLAXO GROUP LIMITED (GB) 2009-05-05 US disclosed
US-7528151-B2 Heterocyclic urea derivatives for the treatment of pain GLAXO GROUP LIMITED (GB) 2009-05-05 US disclosed